CCBE1 promotes GIST development through enhancing angiogenesis and mediating resistance to imatinib

Sci Rep. 2016 Aug 10:6:31071. doi: 10.1038/srep31071.

Abstract

Gastrointestinal stromal tumor (GIST) is the most major mesenchymal neoplasm of the digestive tract. Up to now, imatinib mesylate has been used as a standard first-line treatment for irresectable and metastasized GIST patients or adjuvant treatment for advanced GIST patients who received surgical resection. However, secondary resistance to imatinib usually happens, resulting in a major obstacle in GIST successful therapy. In this study, we first found that collagen and calcium binding EGF domains 1 (CCBE1) expression gradually elevated along with the risk degree of NIH classification, and poor prognosis emerged in the CCBE1-positive patients. In vitro experiments showed that recombinant CCBE1 protein can enhance angiogenesis and neutralize partial effect of imatinib on the GIST-T1 cells. In conclusion, these data indicated that CCBE1 may be served as a new predictor of prognosis in post-operative GIST patients and may play an important role in stimulating GIST progression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents / therapeutic use*
  • Calcium-Binding Proteins / genetics
  • Calcium-Binding Proteins / metabolism*
  • Carcinogenesis
  • Cell Line, Tumor
  • Drug Resistance
  • Female
  • Gastrointestinal Stromal Tumors / drug therapy
  • Gastrointestinal Stromal Tumors / metabolism*
  • Gastrointestinal Stromal Tumors / mortality
  • Gene Expression Regulation, Neoplastic
  • Humans
  • Imatinib Mesylate / therapeutic use*
  • Male
  • Middle Aged
  • Neovascularization, Pathologic
  • Prognosis
  • Survival Analysis
  • Tumor Suppressor Proteins / genetics
  • Tumor Suppressor Proteins / metabolism*
  • Up-Regulation

Substances

  • Antineoplastic Agents
  • CCBE1 protein, human
  • Calcium-Binding Proteins
  • Tumor Suppressor Proteins
  • Imatinib Mesylate