Hemolysis after Oral Artemisinin Combination Therapy for Uncomplicated Plasmodium falciparum Malaria

Emerg Infect Dis. 2016 Aug;22(8):1381-6. doi: 10.3201/eid2208.151905.

Abstract

Episodes of delayed hemolysis 2-6 weeks after treatment of severe malaria with intravenous artesunate have been described. We performed a prospective observational study of patients with uncomplicated malaria to investigate whether posttreatment hemolysis also occurs after oral artemisinin-based combination therapy. Eight of 20 patients with uncomplicated malaria who were given oral artemisinin-based combination therapy met the definition of posttreatment hemolysis (low haptoglobin level and increased lactate dehydrogenase level on day 14). Five patients had hemolysis persisting for 1 month. Patients with posttreatment hemolysis had a median decrease in hemoglobin level of 1.3 g/dL (interquartile range 0.3-2.0 g/dL) in the posttreatment period, and patients without posttreatment hemolysis had a median increase of 0.3 g/dL (IQR -0.1 to 0.7 g/dL; p = 0.002). These findings indicate a need for increased vigilance for hemolytic events in malaria patients, particularly those with predisposing factors for anemia.

Keywords: Plasmodium falciparum; anemia; artemisinin; clinical study; haptoglobin; hemoglobin; hemolysis; lactate dehydrogenase; malaria; oral artemisinin combination therapy; parasites; uncomplicated malaria.

Publication types

  • Observational Study

MeSH terms

  • Administration, Oral
  • Adolescent
  • Adult
  • Anemia / chemically induced
  • Antimalarials / administration & dosage
  • Antimalarials / adverse effects
  • Antimalarials / therapeutic use
  • Artemether
  • Artemisinins / administration & dosage
  • Artemisinins / adverse effects*
  • Artemisinins / therapeutic use*
  • Child
  • Drug Therapy, Combination
  • Ethanolamines / administration & dosage
  • Ethanolamines / therapeutic use
  • Female
  • Fluorenes / administration & dosage
  • Fluorenes / therapeutic use
  • Hemolysis / drug effects*
  • Humans
  • Lumefantrine
  • Malaria, Falciparum / drug therapy*
  • Male
  • Prospective Studies
  • Quinolines / administration & dosage
  • Quinolines / therapeutic use

Substances

  • Antimalarials
  • Artemisinins
  • Ethanolamines
  • Fluorenes
  • Quinolines
  • artenimol
  • piperaquine
  • Artemether
  • Lumefantrine