9-Fluorenylmethyl (Fm) Disulfides: Biomimetic Precursors for Persulfides

Org Lett. 2016 Mar 4;18(5):904-7. doi: 10.1021/acs.orglett.5b03557. Epub 2016 Feb 12.

Abstract

The development of a functional disulfide, FmSSPy-A (Fm = 9-fluorenylmethyl; Py = pyridinyl), is reported. It can effectively convert small molecule and protein thiols (-SH) to form -S-SFm adducts under mild conditions. This method allows for a H2S-free and biomimetic protocol to generate highly reactive persulfides (in their anionic forms). The high nucleophilicity of persulfides toward a number of thiol-blocking reagents is also demonstrated. The method holds promise for further understanding the chemical biology of persulfides and S-sulfhydration.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Biomimetics
  • Disulfides / chemistry*
  • Fluorenes / chemistry*
  • Molecular Structure
  • Sulfides / chemistry*

Substances

  • Disulfides
  • Fluorenes
  • Sulfides
  • persulfides