RelA-Induced Interferon Response Negatively Regulates Proliferation

PLoS One. 2015 Oct 13;10(10):e0140243. doi: 10.1371/journal.pone.0140243. eCollection 2015.

Abstract

Both oncogenic and tumor-suppressor activities are attributed to the Nuclear Factor kappa B (NF-kB) pathway. Moreover, NF-kB may positively or negatively regulate proliferation. The molecular determinants of these opposing roles of NF-kB are unclear. Using primary human mammary epithelial cells (HMEC) as a model, we show that increased RelA levels and consequent increase in basal transcriptional activity of RelA induces IRF1, a target gene. Induced IRF1 upregulates STAT1 and IRF7, and in consort, these factors induce the expression of interferon response genes. Activation of the interferon pathway down-regulates CDK4 and up-regulates p27 resulting in Rb hypo-phosphorylation and cell cycle arrest. Stimulation of HMEC with IFN-γ elicits similar phenotypic and molecular changes suggesting that basal activity of RelA and IFN-γ converge on IRF1 to regulate proliferation. The anti-proliferative RelA-IRF1-CDK4 signaling axis is retained in ER+/HER2- breast tumors analyzed by The Cancer Genome Atlas (TCGA). Using immuno-histochemical analysis of breast tumors, we confirm the negative correlation between RelA levels and proliferation rate in ER+/HER2- breast tumors. These findings attribute an anti-proliferative tumor-suppressor role to basal RelA activity. Inactivation of Rb, down-regulation of RelA or IRF1, or upregulation of CDK4 or IRF2 rescues the RelA-IRF1-CDK4 induced proliferation arrest in HMEC and are points of disruption in aggressive tumors. Activity of the RelA-IRF1-CDK4 axis may explain favorable response to CDK4/6 inhibition observed in patients with ER+ Rb competent tumors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Breast / cytology
  • Breast Neoplasms / pathology
  • Cell Cycle Checkpoints / drug effects
  • Cell Line
  • Cell Proliferation / drug effects
  • Cyclin-Dependent Kinase 4 / metabolism
  • Down-Regulation / drug effects
  • Epithelial Cells / cytology
  • Fallopian Tubes / cytology
  • Female
  • Humans
  • Interferon Regulatory Factor-1 / metabolism
  • Interferon-gamma / metabolism
  • Interferons / pharmacology*
  • MicroRNAs / metabolism
  • Phosphorylation / drug effects
  • Retinoblastoma Protein / metabolism
  • Transcription Factor RelA / metabolism*
  • Tumor Suppressor Protein p53 / metabolism

Substances

  • IRF1 protein, human
  • Interferon Regulatory Factor-1
  • MicroRNAs
  • Retinoblastoma Protein
  • Transcription Factor RelA
  • Tumor Suppressor Protein p53
  • Interferon-gamma
  • Interferons
  • Cyclin-Dependent Kinase 4

Associated data

  • GEO/GSE65040