Plasma apolipoprotein H limits HCV replication and associates with response to NS3 protease inhibitors-based therapy

Liver Int. 2015 Jul;35(7):1833-44. doi: 10.1111/liv.12759. Epub 2015 Jan 23.

Abstract

Background & aims: Chronic infection with HCV remains a public health problem with approximately 150 million people infected worldwide. HCV intersects with lipid metabolism for replication and entry; and plasma concentrations of apolipoproteins have been identified as predictors for response to therapy. Herein, we conducted a screen of plasma proteins, including all apolipoproteins, to identify correlates of response to pegylated-interferon/ribavirin (PR) and HCV non-structural protein 3 (NS3) inhibitors (i.e., telaprevir/boceprevir) therapy in treatment-experienced cirrhotic patients from the ANRS CUPIC cohort.

Methods: We analysed 220 baseline plasma protein concentrations in 189 patients using Luminex technology and analyzed results.

Results: We identified baseline levels of apolipoprotein H (apoH) as a surrogate marker for sustained virological response (SVR). Notably, increased plasma concentration of apoH, used in combination with known clinical parameters, established a robust model with improved classification of patients as likely to achieve SVR (AUC = 0.77, Se = 66%, Sp = 72%, NRI = 39%). Moreover, we provide mechanistic information that indicates a previously unidentified role for apoH during viral entry. Using a human liver slices HCV infection model, we demonstrate that apoH limits replication.

Conclusion: These data support testing of new biomarker strategies for the management of cirrhotic HCV patients and expand our understanding of how apoH may intersect with HCV infection.

Trial registration: ClinicalTrials.gov NCT01514890.

Keywords: HCV protease inhibitor; apolipoprotein H; biomarker; chronic hepatitis C; virological response.

Publication types

  • Clinical Trial
  • Multicenter Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Antiviral Agents / therapeutic use*
  • Area Under Curve
  • Biomarkers / blood
  • Drug Therapy, Combination
  • Female
  • France
  • Hepacivirus / drug effects*
  • Hepacivirus / enzymology
  • Hepacivirus / genetics
  • Hepacivirus / growth & development
  • Hepatitis C, Chronic / blood
  • Hepatitis C, Chronic / diagnosis
  • Hepatitis C, Chronic / drug therapy*
  • Humans
  • Interferon-alpha / therapeutic use
  • Male
  • Middle Aged
  • Molecular Targeted Therapy
  • Oligopeptides / therapeutic use
  • Polyethylene Glycols / therapeutic use
  • Predictive Value of Tests
  • Proline / analogs & derivatives
  • Proline / therapeutic use
  • Prospective Studies
  • Protease Inhibitors / therapeutic use*
  • RNA, Viral / blood
  • ROC Curve
  • Recombinant Proteins / therapeutic use
  • Ribavirin / therapeutic use
  • Time Factors
  • Treatment Outcome
  • Viral Load
  • Viral Nonstructural Proteins / antagonists & inhibitors*
  • Viral Nonstructural Proteins / metabolism
  • Virus Replication / drug effects*
  • beta 2-Glycoprotein I / blood*

Substances

  • Antiviral Agents
  • Biomarkers
  • Interferon-alpha
  • NS3 protein, hepatitis C virus
  • Oligopeptides
  • Protease Inhibitors
  • RNA, Viral
  • Recombinant Proteins
  • Viral Nonstructural Proteins
  • beta 2-Glycoprotein I
  • Polyethylene Glycols
  • Ribavirin
  • telaprevir
  • N-(3-amino-1-(cyclobutylmethyl)-2,3-dioxopropyl)-3-(2-((((1,1-dimethylethyl)amino)carbonyl)amino)-3,3-dimethyl-1-oxobutyl)-6,6-dimethyl-3-azabicyclo(3.1.0)hexan-2-carboxamide
  • Proline
  • peginterferon alfa-2a

Associated data

  • ClinicalTrials.gov/NCT01514890