The effects of ethanol and Ro 15-4513 on elevated plus-maze and rotarod performance in long-sleep and short-sleep mice

Alcohol. 1989 Sep-Oct;6(5):369-76. doi: 10.1016/0741-8329(89)90006-2.

Abstract

The effects of ethanol and diazepam were examined in long-sleep (LS) and short-sleep (SS) mice using the elevated plus-maze. Ethanol had more pronounced effects in SS mice than in LS mice. In contrast, LS mice were more sensitive to the effects of diazepam on the elevated plus-maze. The ataxic effects of ethanol were measured by rotarod performance. SS mice were more resistant to the ataxic effects of a 2.0 g/kg dose of ethanol than LS mice. Ro 15-4513 reversed ethanol's ataxic effects when administered after ethanol in both LS mice and SS mice. Pentobarbital-induced ataxia was unaffected by treatment with Ro 15-4513. Studies of competition of Ro 15-4513 on 3H-flunitrazepam binding indicated that LS and SS mice did not differ in this measure in cortex, cerebellum or hippocampus.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Azides / metabolism
  • Azides / pharmacology*
  • Benzodiazepines / metabolism
  • Benzodiazepines / pharmacology*
  • Binding, Competitive
  • Diazepam / pharmacology
  • Dose-Response Relationship, Drug
  • Ethanol / antagonists & inhibitors
  • Ethanol / pharmacology*
  • Female
  • Flumazenil / pharmacology
  • Flunitrazepam / metabolism
  • Male
  • Mice
  • Mice, Inbred Strains / genetics
  • Motor Activity / drug effects*
  • Sleep / physiology*

Substances

  • Azides
  • Benzodiazepines
  • Ethanol
  • Flumazenil
  • Flunitrazepam
  • Ro 15-4513
  • Diazepam