Differential metabolism of 4-hydroxynonenal in liver, lung and brain of mice and rats

Toxicol Appl Pharmacol. 2014 Aug 15;279(1):43-52. doi: 10.1016/j.taap.2014.04.026. Epub 2014 May 14.

Abstract

The lipid peroxidation end-product 4-hydroxynonenal (4-HNE) is generated in tissues during oxidative stress. As a reactive aldehyde, it forms Michael adducts with nucleophiles, a process that disrupts cellular functioning. Liver, lung and brain are highly sensitive to xenobiotic-induced oxidative stress and readily generate 4-HNE. In the present studies, we compared 4-HNE metabolism in these tissues, a process that protects against tissue injury. 4-HNE was degraded slowly in total homogenates and S9 fractions of mouse liver, lung and brain. In liver, but not lung or brain, NAD(P)+ and NAD(P)H markedly stimulated 4-HNE metabolism. Similar results were observed in rat S9 fractions from these tissues. In liver, lung and brain S9 fractions, 4-HNE formed protein adducts. When NADH was used to stimulate 4-HNE metabolism, the formation of protein adducts was suppressed in liver, but not lung or brain. In both mouse and rat tissues, 4-HNE was also metabolized by glutathione S-transferases. The greatest activity was noted in livers of mice and in lungs of rats; relatively low glutathione S-transferase activity was detected in brain. In mouse hepatocytes, 4-HNE was rapidly taken up and metabolized. Simultaneously, 4-HNE-protein adducts were formed, suggesting that 4-HNE metabolism in intact cells does not prevent protein modifications. These data demonstrate that, in contrast to liver, lung and brain have a limited capacity to metabolize 4-HNE. The persistence of 4-HNE in these tissues may increase the likelihood of tissue injury during oxidative stress.

Keywords: 4-Hydroxynonenal; Alcohol dehydrogenase; Lipid peroxidation; Neurotoxicity; Pulmonary toxicity; Reactive oxygen species.

Publication types

  • Comparative Study
  • Research Support, N.I.H., Extramural

MeSH terms

  • Aldehydes / antagonists & inhibitors
  • Aldehydes / metabolism*
  • Animals
  • Antibodies, Blocking / pharmacology
  • Blotting, Western
  • Brain / drug effects
  • Brain / enzymology
  • Brain / metabolism*
  • Enzyme Inhibitors / pharmacology
  • Glutathione Transferase / antagonists & inhibitors
  • Glutathione Transferase / metabolism
  • Hepatocytes / drug effects
  • Hepatocytes / metabolism
  • Kinetics
  • Liver / drug effects
  • Liver / enzymology
  • Liver / metabolism*
  • Lung / drug effects
  • Lung / enzymology
  • Lung / metabolism*
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Rats
  • Rats, Long-Evans
  • Species Specificity
  • Subcellular Fractions / enzymology
  • Subcellular Fractions / metabolism

Substances

  • Aldehydes
  • Antibodies, Blocking
  • Enzyme Inhibitors
  • Glutathione Transferase
  • 4-hydroxy-2-nonenal