Syndecan-1 (CD138) modulates triple-negative breast cancer stem cell properties via regulation of LRP-6 and IL-6-mediated STAT3 signaling

PLoS One. 2013 Dec 31;8(12):e85737. doi: 10.1371/journal.pone.0085737. eCollection 2013.

Abstract

Syndecan-1 (CD138), a heparan sulfate proteoglycan, acts as a coreceptor for growth factors and chemokines and is a molecular marker associated with epithelial-mesenchymal transition during development and carcinogenesis. Resistance of Syndecan-1-deficient mice to experimentally-induced tumorigenesis has been linked to altered Wnt-responsive precursor cell pools, suggesting a potential role of Syndecan-1 in breast cancer cell stem function. However, the precise molecular mechanism is still elusive. Here, we decipher the functional impact of Syndecan-1 knockdown using RNA interference on the breast cancer stem cell phenotype of human triple-negative MDA-MB-231 and hormone receptor-positive MCF-7 cells in vitro employing an analytical flow cytometric approach. Successful Syndecan-1 siRNA knockdown was confirmed by flow cytometry. Side population measurement by Hoechst dye exclusion and Aldehyde dehydrogenase-1 activity revealed that Syndecan-1 knockdown in MDA-MB-231 cells significantly reduced putative cancer stem cell pools by 60% and 27%, respectively, compared to controls. In MCF-7 cells, Syndecan-1 depletion reduced the side population by 40% and Aldehyde dehydrogenase-1 by 50%, repectively. In MDA-MB-231 cells, the CD44(+)CD24(-/low) phenotype decreased significantly by 6% upon siRNA-mediated Syndecan-1 depletion. Intriguingly, IL-6, its receptor sIL-6R, and the chemokine CCL20, implicated in regulating stemness-associated pathways, were downregulated by >40% in Syndecan-1-silenced MDA-MB-231 cells, which showed a dysregulated response to IL-6-induced shifts in E-cadherin and vimentin expression. Furthermore, activation of STAT-3 and NFkB transcription factors and expression of a coreceptor for Wnt signaling, LRP-6, were reduced by >45% in Syndecan-1-depleted cells compared to controls. At the functional level, Syndecan-1 siRNA reduced the formation of spheres and cysts in MCF-7 cells grown in suspension culture. Our study demonstrates the viability of flow cytometric approaches in analyzing cancer stem cell function. As Syndecan-1 modulates the cancer stem cell phenotype via regulation of the Wnt and IL-6/STAT3 signaling pathways, it emerges as a promising novel target for therapeutic approaches.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aldehyde Dehydrogenase 1 Family
  • Cell Differentiation
  • Down-Regulation
  • Gene Knockdown Techniques
  • Gene Silencing
  • Humans
  • Interleukin-6 / metabolism*
  • Isoenzymes / metabolism
  • Low Density Lipoprotein Receptor-Related Protein-6 / metabolism*
  • MCF-7 Cells
  • NF-kappa B / metabolism
  • Neoplastic Stem Cells / pathology*
  • RNA, Small Interfering / genetics
  • Retinal Dehydrogenase / metabolism
  • STAT3 Transcription Factor / metabolism*
  • Signal Transduction*
  • Spheroids, Cellular / pathology
  • Syndecan-1 / deficiency
  • Syndecan-1 / genetics
  • Syndecan-1 / metabolism*
  • Triple Negative Breast Neoplasms / pathology*
  • Wnt Proteins / metabolism

Substances

  • Interleukin-6
  • Isoenzymes
  • LRP6 protein, human
  • Low Density Lipoprotein Receptor-Related Protein-6
  • NF-kappa B
  • RNA, Small Interfering
  • STAT3 Transcription Factor
  • Syndecan-1
  • Wnt Proteins
  • Aldehyde Dehydrogenase 1 Family
  • ALDH1A1 protein, human
  • ALDH1A1 protein, mouse
  • Retinal Dehydrogenase

Grants and funding

This work was supported by German Academic Exchange Service DAAD A/06/90277 (to SAI), DAAD 56808461 Al Tawasul (to MG and SAI), International Research Training Group “Molecular and Cellular GlycoSciences” Grant GRK 1549 (to MG and SKK), and Maria Möller Stiftung (to MG). The funders had no role in study design, data collection and analysis, decision to publish, or preparation of the manuscript.