Sodium and potassium competition in potassium-selective and non-selective channels

Nat Commun. 2013:4:2721. doi: 10.1038/ncomms3721.

Abstract

Potassium channels selectively conduct K(+), primarily to the exclusion of Na(+), despite the fact that both ions can bind within the selectivity filter. Here we perform crystallographic titration and single-channel electrophysiology to examine the competition of Na(+) and K(+) binding within the filter of two NaK channel mutants; one is the potassium-selective NaK2K mutant and the other is the non-selective NaK2CNG, a CNG channel pore mimic. With high-resolution structures of these engineered NaK channel constructs, we explicitly describe the changes in K(+) occupancy within the filter upon Na(+) competition by anomalous diffraction. Our results demonstrate that the non-selective NaK2CNG still retains a K(+)-selective site at equilibrium, whereas the NaK2K channel filter maintains two high-affinity K(+) sites. A double-barrier mechanism is proposed to explain K(+) channel selectivity at low K(+) concentrations.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Bacillus cereus / metabolism
  • Bacillus subtilis / metabolism
  • Bacterial Proteins / metabolism
  • Binding Sites
  • Binding, Competitive
  • Crystallography, X-Ray
  • Electrophysiology
  • Escherichia coli / metabolism
  • Ion Channel Gating*
  • Liposomes / metabolism
  • Mutation
  • Potassium / metabolism*
  • Potassium Channels / metabolism*
  • Protein Conformation
  • Sodium / metabolism*

Substances

  • Bacterial Proteins
  • Liposomes
  • Potassium Channels
  • Sodium
  • Potassium