Fatal measles virus infection prevented by brain-penetrant fusion inhibitors

J Virol. 2013 Dec;87(24):13785-94. doi: 10.1128/JVI.02436-13. Epub 2013 Oct 9.

Abstract

Measles virus (MV) infection causes an acute childhood disease that can include infection of the central nervous system and can rarely progress to severe neurological disease for which there is no specific treatment. We generated potent antiviral peptide inhibitors of MV entry and spreading and MV-induced cell fusion. Dimers of MV-specific peptides derived from the C-terminal heptad repeat region of the MV fusion protein, conjugated to cholesterol, efficiently protect SLAM transgenic mice from fatal MV infection. Fusion inhibitors hold promise for the prophylaxis of MV infection in unvaccinated and immunocompromised people, as well as potential for the treatment of grave neurological complications of measles.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Antiviral Agents / pharmacology*
  • Brain / drug effects
  • Brain / virology*
  • Cell Line
  • Humans
  • Measles / drug therapy
  • Measles / mortality
  • Measles / prevention & control*
  • Measles / virology
  • Measles virus / drug effects*
  • Measles virus / genetics
  • Measles virus / physiology
  • Mice
  • Mice, Transgenic
  • Viral Fusion Proteins / antagonists & inhibitors*
  • Viral Fusion Proteins / genetics
  • Viral Fusion Proteins / metabolism
  • Virus Internalization / drug effects

Substances

  • Antiviral Agents
  • Viral Fusion Proteins