Stereocontrolled synthesis of 1,3-diols from enones: cooperative Lewis base-mediated intramolecular carbonyl hydrosilylations

J Org Chem. 2013 Sep 20;78(18):9093-101. doi: 10.1021/jo401293a. Epub 2013 Sep 6.

Abstract

A streamlined synthesis of β-hydroxy ketone substrates has been developed to further investigate a recently discovered cooperative Lewis base-mediated intramolecular carbonyl hydrosilylation reaction. The synthesis features an enone β-borylation/oxidation sequence that has proven to be quite general and high-yielding. This has allowed for additional investigations into the diastereoselectivity of the hydrosilylation reaction through the preparation of important polyketide fragments.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Alcohols / chemical synthesis*
  • Alcohols / chemistry
  • Ketones / chemistry*
  • Lewis Bases / chemistry*
  • Molecular Structure
  • Silanes / chemical synthesis
  • Silanes / chemistry*
  • Stereoisomerism

Substances

  • Alcohols
  • Ketones
  • Lewis Bases
  • Silanes