p55PIK-PI3K stimulates angiogenesis in colorectal cancer cell by activating NF-κB pathway

Angiogenesis. 2013 Jul;16(3):561-73. doi: 10.1007/s10456-013-9336-y. Epub 2013 Jan 26.

Abstract

Vascular growth factor (VEGF) is an important mediator of angiogenesis. PI3K plays essential roles in angiogenesis; however, the mechanisms and specific functions of individual isoforms of PI3K members in tumor angiogenesis regulation are still not fully understood. In this study, we evaluate the role of p55PIK, a PI3K regulatory subunit encoded by PIK3R3 gene, in tumor angiogenesis. We reported that overexpression of p55PIK in cancer cells up-regulated HIF-1α expression and increased VEGF expression. Furthermore, overexpression of p55PIK increased tumor angiogenesis in vivo and in vitro. Moreover, data indicated enhanced HIF-1α expression by p55PIK-PI3K depended on its ability to activate NF-кB signaling pathways, especially to increase the phosphorylation of p65 subunits of NF-κB. Our study suggested that p55PIK-PI3K was essential in regulating cancer cell-mediated angiogenesis and contributed to tumor growth and that the p55PIK provides a potential and specific target for new anti-angiogenesis drug development.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Blotting, Western
  • Cell Line, Tumor
  • Colorectal Neoplasms / physiopathology*
  • DNA Primers / genetics
  • Gene Expression Regulation, Neoplastic / physiology*
  • Human Umbilical Vein Endothelial Cells
  • Humans
  • Hypoxia-Inducible Factor 1, alpha Subunit / metabolism
  • Microarray Analysis
  • NF-kappa B / metabolism*
  • Neovascularization, Pathologic / physiopathology*
  • Phosphatidylinositol 3-Kinases / metabolism*
  • Real-Time Polymerase Chain Reaction
  • Signal Transduction / physiology*
  • Vascular Endothelial Growth Factor A / metabolism

Substances

  • DNA Primers
  • HIF1A protein, human
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • NF-kappa B
  • Vascular Endothelial Growth Factor A
  • Phosphatidylinositol 3-Kinases
  • PIK3R3 protein, human