SDF-1α upregulation by atorvastatin in rats with acute myocardial infarction via nitric oxide production confers anti-inflammatory and anti-apoptotic effects

J Biomed Sci. 2012 Nov 21;19(1):99. doi: 10.1186/1423-0127-19-99.

Abstract

Background: The effects of atorvastatin on SDF-1α expression under acute myocardial infarction (AMI) are still unclear. Therefore, our present study is to investigate the roles and mechanisms of atorvastatin treatment on SDF-1α expression in rats with AMI.

Methods: Male Sprague-Dawley rats were underwent permanent coronary artery ligation and randomly assigned into four groups as follow: blank control (B), atorvastatin (A), atorvastatin plus L-NAME (A+L-NAME), and atorvastatin plus AMD3100 (A+AMD3100). Rats underwent similar procedure but without ligation were used as group sham operated (S). Atorvastatin (10mg/Kg/d body weight) was administrated by gavage to rats in three atorvastatin treated groups, and L-NAME (40 mg/Kg/d body weight) or AMD3100 (5mg/Kg/d body weight) was given to group A+L-NAME or A+AMD3100, respectively.

Results: Comparing with group B, NO production, SDF-1α and CXCR4 expression were significantly up-regulated in three atorvastatin treated groups at the seventh day. However, the increments of SDF-1α and CXCR4 expression in group A+L-NAME were reduced when NO production was inhibited by L-NAME. Anti-inflammatory and anti-apoptotic effects of atorvastatin were offset either by decrease of SDF-1α and CXCR4 expression (by L-NAME) or blockage of SDF-1α coupling with CXCR4 (by AMD3100). Expression of STAT3, a cardioprotective factor mediating SDF-1α/CXCR4 axis induced cardiac protection, was up-regulated most significantly in group A. The effects of atorvastatin therapy on cardiac function were also abrogated either when SDF-1α and CXCR4 expression was diminished or the coupling of SDF-1α with CXCR4 was blocked.

Conclusion: SDF-1α upregulation by atorvastatin in rats with AMI was, at least partially, via the eNOS/NO dependent pathway, and SDF-1α upregulation and SDF-1α coupling with CXCR4 conferred anti-inflammatory and anti-apoptotic effects under AMI setting which we speculated that ultimately contributed to cardiac function improvement.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / administration & dosage
  • Apoptosis* / drug effects
  • Atorvastatin
  • Benzylamines
  • Chemokine CXCL12* / genetics
  • Chemokine CXCL12* / metabolism
  • Coronary Vessels / surgery
  • Cyclams
  • Heptanoic Acids* / administration & dosage
  • Heterocyclic Compounds / administration & dosage
  • Ligation / methods
  • Male
  • Myocardial Infarction* / drug therapy
  • Myocardial Infarction* / metabolism
  • Myocardial Infarction* / physiopathology
  • NG-Nitroarginine Methyl Ester / administration & dosage
  • Nitric Oxide* / biosynthesis
  • Nitric Oxide* / metabolism
  • Pyrroles* / administration & dosage
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, CXCR4 / genetics
  • Receptors, CXCR4 / metabolism
  • STAT3 Transcription Factor / metabolism
  • Up-Regulation / drug effects

Substances

  • Anti-Inflammatory Agents
  • Benzylamines
  • Chemokine CXCL12
  • Cxcr4 protein, rat
  • Cyclams
  • Heptanoic Acids
  • Heterocyclic Compounds
  • Pyrroles
  • Receptors, CXCR4
  • STAT3 Transcription Factor
  • Stat3 protein, rat
  • Nitric Oxide
  • Atorvastatin
  • plerixafor
  • NG-Nitroarginine Methyl Ester