Inhibitory effect of adenovirus-mediated siRNA-targeting BMPR-IB on UHMWPE-induced bone destruction in the murine air pouch model

Connect Tissue Res. 2012;53(6):528-34. doi: 10.3109/03008207.2012.702817. Epub 2012 Jul 24.

Abstract

Objective: Adenovirus expressing small interfering RNA (siRNA)-targeting BMPR-IB was locally administered into the air pouch of mice to improve bone resorption induced by ultra-high molecular weight polyethylene (UHMWPE) particles.

Method: Air pouches were established on the back of BALB/c mice, followed by the surgical introduction of a section of calvaria from a syngeneic mouse donor. The bone-implanted pouches were stimulated with the UHMWPE suspension. UHMWPE-containing mice were divided into three study groups to receive injections of adenovirus expressing BMPR-IB siRNA (BMPR-IB group), adenovirus expressing missense siRNA, and virus-free culture medium (control group) into the pouches, respectively. The tissues were harvested at 14 days after the treatment for molecular and histological analyses.

Results: Adenovirus-mediated BMPR-IB siRNA treatment significantly improved UHMWPE particle-induced bone resorption, reduced TRAP and RANK gene and protein expression levels, and diminished the number of TRAP-positive cells. Furthermore, the BMPR-IB siRNA inhibited osteoclast differentiation by targeting osteoblast for the induction of osteoprotegerin formation and downregulation of receptor for activation of nuclear factor-κB ligand production.

Conclusions: This study suggested that loss of bone morphogenetic protein signaling by BMPR-IB siRNA directs osteoblasts to decrease bone destruction in part by downregulating osteoclastogenesis through the receptor for activation of nuclear factor-κB ligand-osteoprotegerin pathway. Local administration of adenovirus expressing siRNA-targeting BMPR-IB may be a feasible and effective therapeutic candidate to treat or prevent wear debris-associated osteolysis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenoviridae*
  • Animals
  • Bone Morphogenetic Protein Receptors, Type I / biosynthesis*
  • Bone Morphogenetic Protein Receptors, Type I / genetics
  • Bone Resorption / chemically induced
  • Bone Resorption / genetics
  • Bone Resorption / metabolism*
  • Bone Resorption / pathology
  • Bone Transplantation
  • Disease Models, Animal
  • Gene Silencing
  • Genetic Vectors*
  • Mice
  • Mice, Inbred BALB C
  • Osteoprotegerin / genetics
  • Osteoprotegerin / metabolism
  • Polyethylene / adverse effects*
  • Polyethylene / pharmacology
  • RNA, Small Interfering*
  • Signal Transduction / drug effects
  • Signal Transduction / genetics
  • Transplantation, Isogeneic

Substances

  • Osteoprotegerin
  • RNA, Small Interfering
  • Tnfrsf11b protein, mouse
  • Polyethylene
  • Bmpr1b protein, mouse
  • Bone Morphogenetic Protein Receptors, Type I