Effects of levosimendan on TNF-alpha, BNP and MMP-1 in patients with heart failure with anemia

Arq Bras Cardiol. 2012 Jul;99(1):659-64. doi: 10.1590/s0066-782x2012005000055. Epub 2012 Jun 26.
[Article in English, Portuguese]

Abstract

Background: Levosimendan is known with its two-sided effects of strengthening myofibril contraction without increasing myocardial oxygen demand. Anemia is a deteriorating situation that causes increase of drug dosing in patients with heart failure.

Objectives: In this study, we compared the effectiveness of levosimendan treatment in decompensated heart failure patients with or without anemia.

Methods: Twenty-three anemic patients having class 3 or 4 heart failure according to New York Heart Association (NYHA) and an ejection fraction of below 35% were included to the study. Another 23 patients with the same cardiac diagnosis but without anemia served as control group. Twenty-four hours levosimendan treatment was added to the traditional heart failure treatment of these patients. Samples were taken to measure serum tumor necrotizing factor alpha (TNF-alpha), aminoterminal pro-brain natriuretic peptide (NT-proBNP) and matrix metalloproteinase-1 (MMP-1) levels before and after the administration.

Results: There was no significant difference between serum TNF-alpha and MMP-1 levels before and after the treatment (p>0.05). Although NT-proBNP level decreased in both groups after the treatment this was not statistically significant (p=0.531 and p=0.913 for anemia and control groups respectively). Significant restoration of functional capacity was seen in both groups assessed according to NYHA (p<0.001 and p=0.001 for anemia and control groups respectively).

Conclusion: Levosimendan treatment shows similar effects in heart failure patients with anemia to that of patients without anemia. However, the early effect of this treatment on TNF-alpha, NT-proBNP and MMP-1 levels is not evident. It provides significant improvement in functional capacity without influence from anemia.

MeSH terms

  • Aged
  • Anemia / blood
  • Anemia / drug therapy*
  • Anemia / physiopathology
  • Cardiotonic Agents / pharmacology
  • Cardiotonic Agents / therapeutic use
  • Chi-Square Distribution
  • Female
  • Heart Failure / blood
  • Heart Failure / drug therapy*
  • Heart Failure / physiopathology
  • Humans
  • Hydrazones / pharmacology
  • Hydrazones / therapeutic use*
  • Infusions, Intravenous
  • Male
  • Matrix Metalloproteinase 1 / blood*
  • Middle Aged
  • Natriuretic Peptide, Brain / blood*
  • Pyridazines / pharmacology
  • Pyridazines / therapeutic use*
  • Simendan
  • Statistics, Nonparametric
  • Treatment Outcome
  • Tumor Necrosis Factor-alpha / blood*

Substances

  • Cardiotonic Agents
  • Hydrazones
  • Pyridazines
  • Tumor Necrosis Factor-alpha
  • Natriuretic Peptide, Brain
  • Simendan
  • Matrix Metalloproteinase 1