Loss of FXR protects against diet-induced obesity and accelerates liver carcinogenesis in ob/ob mice

Mol Endocrinol. 2012 Feb;26(2):272-80. doi: 10.1210/me.2011-1157. Epub 2012 Jan 19.

Abstract

Farnesoid X receptor (FXR) is known to play important regulatory roles in bile acid, lipid, and carbohydrate metabolism. Aged (>12 months old) Fxr(-/-) mice also develop spontaneous liver carcinomas. In this report, we used three mouse models to investigate the role of FXR deficiency in obesity. As compared with low-density lipoprotein receptor (Ldlr) knockout (Ldlr(-/-)) mice, the Ldlr(-/-)Fxr(-/-) double-knockout mice were highly resistant to diet-induced obesity, which was associated with increased expression of genes involved in energy metabolism in the skeletal muscle and brown adipose tissue. Such a striking effect of FXR deficiency on obesity on an Ldlr(-/-) background led us to investigate whether FXR deficiency alone is sufficient to affect obesity. As compared with wild-type mice, Fxr(-/-) mice showed resistance to diet-induced weight gain. Interestingly, only female Fxr(-/-) mice showed significant resistance to diet-induced obesity, which was accompanied by increased energy expenditure in these mice. Finally, we determined the effect of FXR deficiency on obesity in a genetically obese and diabetic mouse model. We generated ob(-/-)Fxr(-/-) mice that were deficient in both Leptin and Fxr. On a chow diet, ob(-/-)Fxr(-/-) mice gained less body weight and had reduced body fat mass as compared with ob/ob mice. In addition, we observed liver carcinomas in 43% of young (<11 months old) Ob(-/-)Fxr(-/-) mice. Together these data indicate that loss of FXR prevents diet-induced or genetic obesity and accelerates liver carcinogenesis under diabetic conditions.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adipose Tissue, Brown / pathology
  • Adiposity / genetics
  • Animals
  • Carcinoma / etiology
  • Carcinoma / genetics*
  • Cell Transformation, Neoplastic / genetics
  • Diet, High-Fat / adverse effects*
  • Dietary Fats / metabolism
  • Energy Metabolism / genetics
  • Female
  • Gene Knockout Techniques
  • Glucose Intolerance / complications
  • Glucose Intolerance / genetics
  • Intestinal Absorption
  • Leptin / deficiency
  • Leptin / genetics
  • Liver / pathology
  • Liver Neoplasms / etiology
  • Liver Neoplasms / genetics*
  • Male
  • Mice
  • Mice, Knockout
  • Mice, Obese
  • Muscle, Skeletal / metabolism
  • Obesity / etiology*
  • Obesity / genetics
  • Receptors, Cytoplasmic and Nuclear / deficiency*
  • Receptors, Cytoplasmic and Nuclear / genetics
  • Sex Factors
  • Weight Gain / genetics

Substances

  • Dietary Fats
  • Leptin
  • Receptors, Cytoplasmic and Nuclear
  • farnesoid X-activated receptor