Sharpin contributes to TNFα dependent NFκB activation and anti-apoptotic signalling in hepatocytes

PLoS One. 2012;7(1):e29993. doi: 10.1371/journal.pone.0029993. Epub 2012 Jan 9.

Abstract

TNFα stimulates both pro- and anti-apoptotic signalling in hepatocytes. Anti-apoptotic signalling depends on a cascade of ubiquitylation steps leading to NFκB activation. Using Sharpin-deficient mice, we show that the ubiquitin binding protein Sharpin interacts with Hoip, an E3 ligase which generates linear ubiquitin chains. Sharpin-deficiency sensitized hepatocytes to induction of apoptosis by TNFα even in the absence of transcriptional inhibition. TNFα induced activation of NFκB was strongly reduced in hepatocytes from Sharpin-deficient mice, due to reduced and delayed phosphorylation and degradation of IκBα. Injection of TNFα-inducing lipopolysaccharides led to strongly exacerbated liver damage and premature death in Sharpin-deficient mice. Our findings point to an essential role of Sharpin in linear ubiquitin chain formation, NFκB activation, and protection of the liver against inflammatory damaging signals.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis / drug effects*
  • Gene Expression Profiling
  • Hepatocytes / drug effects*
  • Hepatocytes / metabolism*
  • Humans
  • Lipopolysaccharides / pharmacology
  • Liver Failure / metabolism
  • Liver Failure / pathology
  • Mice
  • Mice, Inbred C57BL
  • NF-kappa B / metabolism*
  • Nerve Tissue Proteins / metabolism*
  • Organ Specificity / drug effects
  • Organ Specificity / genetics
  • Protein Binding / drug effects
  • Rats
  • Signal Transduction / drug effects*
  • Tumor Necrosis Factor-alpha / pharmacology*
  • Ubiquitin / metabolism
  • Ubiquitin-Protein Ligases / metabolism

Substances

  • Lipopolysaccharides
  • NF-kappa B
  • Nerve Tissue Proteins
  • Tumor Necrosis Factor-alpha
  • Ubiquitin
  • sharpin
  • Rnf31 protein, mouse
  • Ubiquitin-Protein Ligases