Time-correlated single photon counting for simultaneous monitoring of zinc oxide nanoparticles and NAD(P)H in intact and barrier-disrupted volunteer skin

Pharm Res. 2011 Nov;28(11):2920-30. doi: 10.1007/s11095-011-0515-5. Epub 2011 Jun 30.

Abstract

Purpose: There is a lack of relevant, non-animal alternatives for assessing exposure and toxicity of nanoparticle-containing cosmetics, e.g. sunscreens. Our goal was to evaluate timecorrelated single photon counting (TCSPC) for simultaneous monitoring of zinc oxide nanoparticles (ZnO-NP) and the metabolic state of volunteer skin.

Methods: We separated the fluorescence lifetime signatures of endogenous fluorophore signals (i.e. nicotinamide adenine dinucleotide phosphate, NAD(P)H and keratin) and the ZnO-NP signal using advanced TCSPC to simultaneously determine ZnO-NP penetration profiles and NAD(P)H changes in subjects with altered barrier function, including tape-stripped skin and in psoriasis or atopic dermatitis lesions.

Results: We detected no ZnO-NP penetration into viable human skin in any group. ZnO-NP signal was significantly increased (p < 0.01) on the surface of tape-stripped and lesional skin after 4 and 2 h of treatment, respectively. Free NAD(P)H signal significantly increased in tape-stripped viable epidermis treated for 4 h of ZnO-NP compared to vehicle control. No significant NAD(P)H changes were noted in the lesional study.

Conclusion: TCSPC techniques enabled simultaneous, real-time quantification of ZnO-NP concentration and NAD(P)H via non-invasive imaging in the stratum corneum and viable epidermis of volunteers.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Administration, Topical
  • Cosmetics / metabolism
  • Dermatitis, Atopic / drug therapy
  • Dermatitis, Atopic / metabolism*
  • Dose-Response Relationship, Drug
  • Drug Delivery Systems*
  • Humans
  • Metal Nanoparticles / administration & dosage
  • Metal Nanoparticles / analysis*
  • Metal Nanoparticles / therapeutic use
  • NADP / analysis*
  • NADP / metabolism
  • Photons
  • Psoriasis / drug therapy
  • Psoriasis / metabolism*
  • Skin / chemistry*
  • Skin / metabolism
  • Skin Absorption
  • Sunscreening Agents / administration & dosage
  • Sunscreening Agents / analysis
  • Sunscreening Agents / metabolism
  • Sunscreening Agents / therapeutic use
  • Surgical Tape
  • Time Factors
  • Toxicity Tests / methods
  • Water Loss, Insensible / physiology
  • Zinc Oxide / administration & dosage
  • Zinc Oxide / analysis
  • Zinc Oxide / metabolism*
  • Zinc Oxide / therapeutic use

Substances

  • Cosmetics
  • Sunscreening Agents
  • NADP
  • Zinc Oxide