Role of cysteine residues in ribonuclease H from Escherichia coli. Site-directed mutagenesis and chemical modification

Biochem J. 1990 Oct 1;271(1):59-66. doi: 10.1042/bj2710059.

Abstract

The role of the three cysteine residues at positions 13, 63 and 133 in Escherichia coli RNAase H, an enzyme that is sensitive to N-ethylmaleimide [Berkower, Leis & Hurwitz (1973) J. Biol. Chem. 248, 5914-5921], was examined by using both site-directed mutagenesis and chemical modification. Novel aspects that were found are as follows. First, none of the cysteine residues is required for activity. Secondly, chemical modification of either Cys-13 or Cys-133 with thiol-blocking reagents inactivates the enzyme, but that of Cys-63 does not. Thus the sensitivity of E. coli RNAase H to N-ethylmaleimide arises not from blocking of the thiol group but from steric hindrance by the modifying group incorporated at either Cys-13 or Cys-133.

MeSH terms

  • Amino Acid Sequence
  • Chemical Phenomena
  • Chemistry
  • Chromatography, High Pressure Liquid
  • Circular Dichroism
  • Cysteine*
  • Dithionitrobenzoic Acid
  • Endoribonucleases / antagonists & inhibitors*
  • Endoribonucleases / chemistry
  • Endoribonucleases / metabolism
  • Escherichia coli / enzymology*
  • Ethylmaleimide / pharmacology*
  • Iodoacetates / pharmacology
  • Iodoacetic Acid
  • Molecular Sequence Data
  • Mutagenesis, Site-Directed*
  • Peptide Mapping
  • Ribonuclease H
  • Serine Endopeptidases / metabolism
  • Structure-Activity Relationship

Substances

  • Iodoacetates
  • Dithionitrobenzoic Acid
  • Endoribonucleases
  • Ribonuclease H
  • Serine Endopeptidases
  • lysyl endopeptidase
  • Cysteine
  • Ethylmaleimide
  • Iodoacetic Acid