Glucose regulates cyclin D2 expression in quiescent and replicating pancreatic β-cells through glycolysis and calcium channels

Endocrinology. 2011 Jul;152(7):2589-98. doi: 10.1210/en.2010-1372. Epub 2011 Apr 26.

Abstract

Understanding the molecular triggers of pancreatic β-cell proliferation may facilitate the development of regenerative therapies for diabetes. Genetic studies have demonstrated an important role for cyclin D2 in β-cell proliferation and mass homeostasis, but its specific function in β-cell division and mechanism of regulation remain unclear. Here, we report that cyclin D2 is present at high levels in the nucleus of quiescent β-cells in vivo. The major regulator of cyclin D2 expression is glucose, acting via glycolysis and calcium channels in the β-cell to control cyclin D2 mRNA levels. Furthermore, cyclin D2 mRNA is down-regulated during S-G(2)-M phases of each β-cell division, via a mechanism that is also affected by glucose metabolism. Thus, glucose metabolism maintains high levels of nuclear cyclin D2 in quiescent β-cells and modulates the down-regulation of cyclin D2 in replicating β-cells. These data challenge the standard model for regulation of cyclin D2 during the cell division cycle and suggest cyclin D2 as a molecular link between glucose levels and β-cell replication.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Calcium Channel Agonists / pharmacology
  • Calcium Channels / metabolism*
  • Cell Cycle
  • Cell Line
  • Cell Nucleus / drug effects
  • Cell Nucleus / metabolism
  • Cell Proliferation*
  • Cyclin D2 / genetics
  • Cyclin D2 / metabolism*
  • Diabetes Mellitus, Experimental / genetics
  • Diabetes Mellitus, Experimental / metabolism
  • Diabetes Mellitus, Experimental / pathology
  • Enzyme Inhibitors / pharmacology
  • Gene Expression Regulation / drug effects
  • Glucose / metabolism*
  • Glycolysis* / drug effects
  • Humans
  • Islets of Langerhans / cytology
  • Islets of Langerhans / drug effects
  • Islets of Langerhans / metabolism*
  • Islets of Langerhans / pathology
  • Male
  • Mice
  • Mice, Inbred ICR
  • Mice, Transgenic
  • Organ Culture Techniques
  • RNA, Messenger / metabolism

Substances

  • CCND2 protein, human
  • Calcium Channel Agonists
  • Calcium Channels
  • Ccnd2 protein, mouse
  • Cyclin D2
  • Enzyme Inhibitors
  • RNA, Messenger
  • Glucose