Cytosolic lysine residues enhance anterograde transport and activation of the erythropoietin receptor

Biochem J. 2011 Apr 15;435(2):509-18. doi: 10.1042/BJ20101876.

Abstract

Lysine residues are key residues in many cellular processes, in part due to their ability to accept a wide variety of post-translational modifications. In the present study, we identify the EPO-R [EPO (erythropoietin) receptor] cytosolic lysine residues as enhancers of receptor function. EPO-R drives survival, proliferation and differentiation of erythroid progenitor cells via binding of its ligand EPO. We mutated the five EPO-R cytosolic lysine residues to arginine residues (5KR EPO-R), eliminating putative lysine-dependent modifications. Overexpressed 5KR EPO-R displayed impaired ubiquitination and improved stability compared with wt (wild-type) EPO-R. Unexpectedly, fusion proteins consisting of VSVGtsO45 (vesicular stomatitis virus glycoprotein temperature-sensitive folding mutant) with wt or 5KR EPO-R cytosolic domains demonstrated delayed glycan maturation kinetics upon substitution of the lysine residues. Moreover, VSVG-wt EPO-R, but not VSVG-5KR EPO-R, displayed endoplasmic reticulum-associated ubiquitination. Despite similar cell-surface EPO-binding levels of both receptors and the lack of EPO-induced ubiquitination by 5KR EPO-R, the lysine-less mutant produced weaker receptor activation and signalling than the wt receptor. We thus propose that EPO-R cytosolic lysine residues enhance receptor function, most probably through ubiquitination and/or other post-translational modifications.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cells, Cultured
  • Cytosol / metabolism
  • Endoplasmic Reticulum / metabolism
  • Humans
  • Lysine / genetics
  • Lysine / metabolism
  • Lysine / physiology*
  • Mice
  • Models, Biological
  • Mutant Proteins / metabolism
  • Protein Processing, Post-Translational / genetics
  • Protein Processing, Post-Translational / physiology
  • Protein Transport / genetics
  • Receptors, Erythropoietin / agonists*
  • Receptors, Erythropoietin / genetics
  • Receptors, Erythropoietin / metabolism*
  • Ubiquitination

Substances

  • Mutant Proteins
  • Receptors, Erythropoietin
  • Lysine