Overexpression of transcription factor sp2 inhibits epidermal differentiation and increases susceptibility to wound- and carcinogen-induced tumorigenesis

Cancer Res. 2010 Nov 1;70(21):8507-16. doi: 10.1158/0008-5472.CAN-10-1213. Epub 2010 Oct 19.

Abstract

Sp proteins are evolutionarily conserved transcription factors required for the expression of a wide variety of genes that are critical for development and cell cycle progression. Deregulated expression of certain Sp proteins is associated with the formation of a variety of human tumors; however, direct evidence that any given Sp protein is oncogenic has been lacking. Here, we report that Sp2 protein abundance in mice increases in concert with the progression of carcinogen-induced murine squamous cell carcinomas. Transgenic mice specifically overexpressing murine Sp2 in epidermal basal keratinocytes were highly susceptible to wound- and carcinogen-induced papillomagenesis. Transgenic animals that were homozygous rather than hemizygous for the Sp2 transgene exhibited a striking arrest in the epidermal differentiation program, perishing within 2 weeks of birth. Our results directly support the likelihood that Sp2 overexpression occurring in various human cancers has significant functional effect.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • 9,10-Dimethyl-1,2-benzanthracene / toxicity*
  • Animals
  • Blotting, Western
  • COS Cells
  • Carcinogens / toxicity
  • Carcinoma, Squamous Cell / etiology
  • Carcinoma, Squamous Cell / metabolism
  • Carcinoma, Squamous Cell / pathology*
  • Cattle
  • Cell Differentiation*
  • Chlorocebus aethiops
  • Disease Susceptibility
  • Epidermal Cells*
  • Epidermis / drug effects
  • Epidermis / metabolism
  • Female
  • Humans
  • Immunoenzyme Techniques
  • Keratin-5 / genetics
  • Keratinocytes / cytology
  • Keratinocytes / drug effects
  • Keratinocytes / metabolism
  • Male
  • Mice
  • Mice, Transgenic
  • Promoter Regions, Genetic
  • RNA, Messenger / genetics
  • Reverse Transcriptase Polymerase Chain Reaction
  • Skin Neoplasms / etiology
  • Skin Neoplasms / metabolism
  • Skin Neoplasms / pathology*
  • Sp2 Transcription Factor / physiology*
  • Wounds and Injuries*

Substances

  • Carcinogens
  • Keratin-5
  • RNA, Messenger
  • Sp2 Transcription Factor
  • 9,10-Dimethyl-1,2-benzanthracene