4F Peptide reduces nascent atherosclerosis and induces natural antibody production in apolipoprotein E-null mice

FASEB J. 2011 Jan;25(1):290-300. doi: 10.1096/fj.10-165670. Epub 2010 Sep 27.

Abstract

Our objective was to contrast the effect of apolipoprotein (apo) A-I mimetic peptides, such as 4F and 4F-Pro-4F (Pro), on nascent and mature atherosclerotic lesions and on levels of antibodies against oxidation-specific epitopes. Chow-fed apoE(-/-) mice were injected intraperitoneally with either the 4F peptide or a tandem helix apoA-I mimetic peptide (Pro) every other day. Mice treated with 4F, but not Pro, for 4 wk starting at 10 wk of age showed a dramatic decrease in atherosclerosis at 2 arterial sites. However, neither peptide was effective in mice treated for 8 wk starting at 20 wk of age; lesions were larger and more mature at this time point. Peptide treatment caused increased production of antibodies against oxidation-specific epitopes, including a disproportionate induction of the IgM natural antibody (NAb) E06/T15 to oxidized phospholipids. In summary, 4F, but not the tandem peptide Pro, effectively inhibited early atherogenesis but was ineffective against more mature lesions. Two different apoA-I mimetic peptides increased titers of natural antibodies against oxidation-specific epitopes.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Age Factors
  • Amino Acid Sequence
  • Animals
  • Antibodies / metabolism*
  • Apolipoprotein A-I / chemistry
  • Apolipoproteins E / deficiency
  • Apolipoproteins E / genetics*
  • Aryldialkylphosphatase / blood
  • Atherosclerosis / blood
  • Atherosclerosis / pathology
  • Atherosclerosis / prevention & control*
  • Body Weight / drug effects
  • Cholesterol, LDL / blood
  • Epitopes / immunology
  • Female
  • Immunoglobulin G / metabolism
  • Immunoglobulin M / metabolism
  • Lipoproteins, LDL / immunology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Molecular Sequence Data
  • Organ Size / drug effects
  • Peptides / chemistry
  • Peptides / pharmacology*
  • Serum Amyloid A Protein / metabolism
  • Spleen / drug effects
  • Spleen / pathology

Substances

  • Antibodies
  • Apolipoprotein A-I
  • Apolipoproteins E
  • Cholesterol, LDL
  • Epitopes
  • Immunoglobulin G
  • Immunoglobulin M
  • Lipoproteins, LDL
  • Peptides
  • Serum Amyloid A Protein
  • oxidized low density lipoprotein
  • Aryldialkylphosphatase