Alanine aminotransferase is an inadequate surrogate marker for detecting lamivudine resistance

World J Gastroenterol. 2010 Oct 7;16(37):4691-6. doi: 10.3748/wjg.v16.i37.4691.

Abstract

Aim: To investigate the accuracy of serum alanine aminotransferase (ALT) in diagnosing lamivudine resistance and factors that contributed to abnormal serum ALT.

Methods: This was a retrospective study of chronic hepatitis B patients on lamivudine therapy who were followed for 3-mo with liver function tests and hepatitis B virus (HBV) DNA measurement. Lamivudine resistance was defined as HBV DNA ≥ 1 log from nadir on at least 2 occasions, confirmed by genotyping. Serum ALT levels in patients with lamivudine resistance were compared to serum ALT levels in those without lamivudine resistance.

Results: There were 111 patients with and 117 without lamivudine resistance. The area under the receiver operating characteristic of serum ALT to diagnose lamivudine resistance was 0.645 ± 0.037. Serum ALT > 42.5 U/L gave the best diagnostic accuracy with sensitivity = 61%, specificity = 60%, positive predictive value = 60%, negative predictive value = 61%, positive likelihood ratio = 1.53 and negative likelihood ratio = 0.65 for predicting lamivudine resistance, missing 39% of resistant patients. Using other serum ALT cutoffs, diagnostic accuracy was lower. By multivariate analysis, baseline abnormal serum ALT was associated with abnormal ALT during resistance (OR = 5.98, P = 0.003), and males were associated with serum ALT flares during resistance (OR = 8.9, P = 0.016).

Conclusion: Serum ALT is inadequate for diagnosing lamivudine resistance and has implications where viral resistance testing is suboptimal and for reimbursement of rescue therapy.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Alanine Transaminase / blood*
  • Antiviral Agents / pharmacology
  • Antiviral Agents / therapeutic use*
  • Asian People
  • Biomarkers / blood*
  • DNA, Viral / blood
  • Drug Resistance, Viral*
  • Hepatitis B virus / drug effects
  • Hepatitis B virus / genetics
  • Hepatitis B, Chronic* / blood
  • Hepatitis B, Chronic* / drug therapy
  • Humans
  • Lamivudine / pharmacology
  • Lamivudine / therapeutic use*
  • Male
  • Middle Aged
  • Retrospective Studies
  • Sensitivity and Specificity

Substances

  • Antiviral Agents
  • Biomarkers
  • DNA, Viral
  • Lamivudine
  • Alanine Transaminase