Drug resistance mutations in HIV-infected patients in the Spanish drug resistance database failing tipranavir and darunavir therapy

Antimicrob Agents Chemother. 2010 Jul;54(7):3018-20. doi: 10.1128/AAC.00160-10. Epub 2010 May 17.

Abstract

The presence of resistance mutations in patients failing tipranavir or darunavir was examined at the national drug resistance database of the Spanish AIDS Research Network. Although mutations emerging during tipranavir and darunavir failures differed considerably, cross-resistance was found in up to half of the patients tested. Interestingly, mutation 54L, which is associated with tipranavir hypersusceptibility, was selected in half of the darunavir failures. Thus, resistance testing seems mandatory to ensure the benefit of the sequential use of these drugs.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Darunavir
  • Databases, Factual*
  • Drug Resistance, Viral / genetics*
  • HIV Infections / drug therapy*
  • HIV Infections / genetics
  • HIV Protease Inhibitors / therapeutic use*
  • Humans
  • Mutation
  • Pyridines / therapeutic use*
  • Pyrones / therapeutic use*
  • Spain
  • Sulfonamides / therapeutic use*

Substances

  • HIV Protease Inhibitors
  • Pyridines
  • Pyrones
  • Sulfonamides
  • Darunavir
  • tipranavir