Diastereoselective Synthesis of trans-beta-Lactams Using a Simple Multifunctional Catalyst

Synlett. 2009:10:1651-1654. doi: 10.1055/s-0029-1217348.

Abstract

A catalytic, highly diastereoselective process for the synthesis of trans-beta-lactams is reported. This system is based on a phosphonium fluoride precatalyst that both activates the nucleophile and directs the reaction process for high yield and diastereoselectivity.