Decreased Beta(2)*-nicotinic acetylcholine receptor availability after chronic ethanol exposure in nonhuman primates

Synapse. 2010 Sep;64(9):729-32. doi: 10.1002/syn.20795.

Abstract

Ethanol associated behaviors have been linked to the beta(2)-subunit containing nicotinic acetylcholine receptors (beta(2)*-nAChR); however, there is conflicting evidence on ethanol-induced changes in nAChR expression during and after chronic ethanol consumption. In this study, five male animals orally self-administered ethanol for 18 +/- 1 weeks. Animals were scanned with [(123)I]5-IA-85380 and SPECT prior to ethanol self-administration, and at 24 h and 5-13 wks withdrawal. beta(2)*-nAChR availability was not significantly different from baseline at 24 h withdrawal, but was significantly decreased compared to baseline at 5-13 wks withdrawal throughout the cortex and in the thalamus, but not the midbrain. The percent decrease in beta(2)*-nAChR availability from baseline to 5-13 wks withdrawal in the parietal cortex was negatively correlated with total grams of ethanol consumed in lifetime and in the midbrain was negatively correlated with average daily ethanol consumption (g/kg). Prolonged withdrawal from chronic ethanol consumption is associated with a decrease in beta(2)*-nAChR availability. The decrease in beta(2)*-nAChR availability is influenced by alcohol consumption, suggesting the chronicity and severity of alcohol consumption may underlie persistent changes in beta(2)*-nAChR availability.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Azetidines
  • Brain / diagnostic imaging
  • Brain Chemistry / drug effects
  • Central Nervous System Depressants / pharmacology
  • Dose-Response Relationship, Drug
  • Ethanol / pharmacology*
  • Linear Models
  • Macaca mulatta
  • Male
  • Pyridines
  • Radiopharmaceuticals
  • Receptors, Nicotinic / drug effects*
  • Receptors, Nicotinic / metabolism*
  • Self Administration
  • Tomography, Emission-Computed, Single-Photon

Substances

  • 5-iodo-3-(2-azetidinylmethoxy)pyridine
  • Azetidines
  • Central Nervous System Depressants
  • Pyridines
  • Radiopharmaceuticals
  • Receptors, Nicotinic
  • nicotinic receptor beta2
  • Ethanol