A role of Miz-1 in Gfi-1-mediated transcriptional repression of CDKN1A

Oncogene. 2010 May 13;29(19):2843-52. doi: 10.1038/onc.2010.48. Epub 2010 Mar 1.

Abstract

Zinc-finger (ZF) transcriptional repressor growth factor independence 1 (Gfi-1) has an important role in hematopoiesis and inner ear development, and also functions as an oncoprotein that cooperates with c-Myc in lymphomagenesis. Gfi-1 represses transcription by directly binding to conserved sequences in the promoters of its target genes. CDKN1A encoding p21(Cip1) has been identified as a Gfi-1 target gene and has been shown to contain Gfi-1 binding sites in the upstream promoter region. We show here that Gfi-1 represses CDKN1A in a manner that is independent of its DNA binding activity. Gfi-1 interacts with POZ-ZF transcription factor Miz-1, originally shown to be a c-Myc-interacting partner, and through Miz-1 binds to the CDKN1A core promoter. Interestingly, Gfi-1 and c-Myc, through Miz-1, form a ternary complex on the CDKN1A promoter, and function in collaboration to repress CDKN1A. Gfi-1 knockdown results in enhanced levels of p21(Cip1) and attenuated cell proliferation. Notably, similar to c-Myc, the expression of Gfi-1 is downregulated by transforming growth factor-beta (TGFbeta) and the level of Gfi-1 influences the response of cells to the cytostatic effect of TGFbeta. Our data reveal an important mechanism by which Gfi-1 regulates cell proliferation and may also have implications for understanding the role of Gfi-1 in lymphomagenesis.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • Cyclin-Dependent Kinase Inhibitor p21 / genetics*
  • Cyclin-Dependent Kinase Inhibitor p21 / metabolism
  • Cytostatic Agents / pharmacology
  • DNA / metabolism
  • DNA-Binding Proteins / chemistry
  • DNA-Binding Proteins / metabolism*
  • Down-Regulation / drug effects
  • Hematopoiesis / drug effects
  • Humans
  • Kruppel-Like Transcription Factors / metabolism*
  • Lymphoma / pathology
  • Mice
  • Promoter Regions, Genetic / genetics
  • Proto-Oncogene Proteins c-myc / metabolism
  • Rats
  • Transcription Factors / chemistry
  • Transcription Factors / metabolism*
  • Transcription, Genetic*
  • Transforming Growth Factor beta / pharmacology
  • Zinc Fingers

Substances

  • Cyclin-Dependent Kinase Inhibitor p21
  • Cytostatic Agents
  • DNA-Binding Proteins
  • Gfi1 protein, rat
  • Kruppel-Like Transcription Factors
  • Proto-Oncogene Proteins c-myc
  • Transcription Factors
  • Transforming Growth Factor beta
  • DNA