Alpha-lipoic acid improves vascular endothelial function in patients with type 2 diabetes: a placebo-controlled randomized trial

Eur J Clin Invest. 2010 Feb;40(2):148-54. doi: 10.1111/j.1365-2362.2009.02236.x. Epub 2009 Dec 27.

Abstract

Objective: The aim of this study was to investigate the effect of alpha-lipoic acid (ALA) treatment on endothelium-dependent and -independent vasodilatation, assessed by forearm blood flow (FBF), in patients with type 2 diabetes mellitus.

Research design and methods: A total of 30 subjects with type 2 diabetes were included in this randomized, controlled, double-blinded, parallel group study. FBF responses to intra-arterial acetylcholine (ACh) and glycerol trinitrate (GTN) were measured before and after 21 days of intravenous treatment with 600 mg alpha-lipoic acid or placebo.

Results: FBF responses were comparable at baseline. After treatment, FBF reactivity to ACh and GTN was unchanged in subjects receiving placebo. By contrast, ALA treatment increased endothelium-dependent vasodilatation to ACh (P < 0.05) but not to GTN compared with baseline.

Conclusions: Intravenous ALA treatment improves endothelium-dependent vasodilatation in patients with type 2 diabetes, in the absence of effects on forearm vasomotor function. If this salutary action translates into vascular risk reduction remains to be established.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylcholine / pharmacology
  • Antioxidants / pharmacology*
  • Antioxidants / therapeutic use
  • Diabetes Mellitus, Type 2 / blood
  • Diabetes Mellitus, Type 2 / drug therapy*
  • Diabetes Mellitus, Type 2 / physiopathology
  • Double-Blind Method
  • Endothelium, Vascular / drug effects*
  • Endothelium, Vascular / physiopathology*
  • Female
  • Forearm / blood supply
  • Forearm / physiopathology
  • Humans
  • Male
  • Middle Aged
  • Nitroglycerin / pharmacology
  • Regional Blood Flow / drug effects
  • Thioctic Acid / pharmacology*
  • Thioctic Acid / therapeutic use
  • Vasodilation / drug effects*
  • Vasodilator Agents / pharmacology*

Substances

  • Antioxidants
  • Vasodilator Agents
  • Thioctic Acid
  • Nitroglycerin
  • Acetylcholine