Phosphorylation-dependent Lys63-linked polyubiquitination of Daxx is essential for sustained TNF-{alpha}-induced ASK1 activation

Cancer Res. 2009 Oct 1;69(19):7512-7. doi: 10.1158/0008-5472.CAN-09-2148. Epub 2009 Sep 29.

Abstract

Apoptosis signal-regulating kinase 1 (ASK1) is a key regulatory kinase in the proapoptotic response to various stresses. ASK1 phosphorylation of Daxx, an ASK1 activator protein, increases Daxx accumulation in cells and further enhances ASK1 activity through a positive feedback mechanism. Here, we show that ASK1-dependent phosphorylation of Daxx induces Lys(63) (K63)-linked polyubiquitination on Lys(122) of Daxx. Polyubiquitination is dispensable for Daxx accumulation or Daxx interaction with ASK1 because mutant Daxx deficient in polyubiquitin still exhibits ASK1-dependent accumulation and interaction with cellular ASK1. However, K63-linked Daxx polyubiquitination is required for tumor necrosis factor-alpha (TNF-alpha)-induced activation of ASK1. Therefore, K63-linked polyubiquitination of Daxx functions as a molecular switch to initiate and amplify the stress kinase response in the TNF-alpha signaling pathway.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adaptor Proteins, Signal Transducing / metabolism*
  • Cell Line, Tumor
  • Co-Repressor Proteins
  • Enzyme Activation
  • HeLa Cells
  • Humans
  • Lysine / metabolism
  • MAP Kinase Kinase Kinase 5 / biosynthesis
  • MAP Kinase Kinase Kinase 5 / genetics
  • MAP Kinase Kinase Kinase 5 / metabolism*
  • Molecular Chaperones
  • Nuclear Proteins / metabolism*
  • Phosphorylation
  • Polyubiquitin / metabolism*
  • Transfection
  • Tumor Necrosis Factor-alpha / metabolism*
  • Ubiquitination

Substances

  • Adaptor Proteins, Signal Transducing
  • Co-Repressor Proteins
  • DAXX protein, human
  • Molecular Chaperones
  • Nuclear Proteins
  • Tumor Necrosis Factor-alpha
  • Polyubiquitin
  • MAP Kinase Kinase Kinase 5
  • MAP3K5 protein, human
  • Lysine