Abstract
The publication of the crystal structures of a bacterial quorum sensing receptor complexed with a variety of ligands (Zou and Nair, 2009) provides a much-needed molecular rationale for the modulation of this intercellular signaling process, which may facilitate the development of new therapeutic agents.
MeSH terms
-
4-Butyrolactone / analogs & derivatives
-
4-Butyrolactone / pharmacology
-
Bacterial Proteins / chemistry*
-
Bacterial Proteins / metabolism
-
Crystallography, X-Ray
-
Protein Binding
-
Pseudomonas aeruginosa / metabolism*
-
Quorum Sensing / physiology*
-
Small Molecule Libraries
-
Terphenyl Compounds / chemistry
-
Terphenyl Compounds / pharmacology*
-
Trans-Activators / chemistry*
-
Trans-Activators / metabolism
Substances
-
Bacterial Proteins
-
LasR protein, Pseudomonas aeruginosa
-
Small Molecule Libraries
-
Terphenyl Compounds
-
Trans-Activators
-
homoserine lactone
-
4-Butyrolactone