Inhibitory effect of somatostatin-14 on L-type voltage-gated calcium channels in cultured cone photoreceptors requires intracellular calcium

J Neurophysiol. 2009 Sep;102(3):1801-10. doi: 10.1152/jn.00354.2009. Epub 2009 Jul 15.

Abstract

The inhibitory effects of somatostatin have been well documented for many physiological processes. The action of somatostatin is through G-protein-coupled receptor-mediated second-messenger signaling, which in turn affects other downstream targets including ion channels. In the retina, somatostatin is released from a specific class of amacrine cells. Here we report that there was a circadian phase-dependent effect of somatostatin-14 (SS14) on the L-type voltage-gated calcium channels (L-VGCCs) in cultured chicken cone photoreceptors, and our study reveals that this process is dependent on intracellular calcium stores. Application of 500 nM SS14 for 2 h caused a decrease in L-VGCC currents only during the subjective night but not the subjective day. We then explored the cellular mechanisms underlying the circadian phase-dependent effect of SS14. The inhibitory effect of SS14 on L-VGCCs was mediated through the pertussis-toxin-sensitive G-protein-dependent somatostatin receptor 2 (sst2). Activation of sst2 by SS14 further activated downstream signaling involving phospholipase C and intracellular calcium stores. Mobilization of intracellular Ca2+ was required for somatostatin induced inhibition of photoreceptor L-VGCCs, suggesting that somatostatin plays an important role in the modulation of photoreceptor physiology.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Calcium / metabolism*
  • Calcium Channels, L-Type / metabolism*
  • Cells, Cultured
  • Chelating Agents / pharmacology
  • Chick Embryo
  • Circadian Rhythm / physiology
  • Cyanamide / metabolism
  • Drug Interactions
  • Egtazic Acid / analogs & derivatives
  • Egtazic Acid / pharmacology
  • Enzyme Inhibitors / pharmacology
  • Gene Expression Regulation / drug effects
  • Hormone Antagonists / pharmacology
  • Hormones / pharmacology*
  • Intracellular Fluid / drug effects*
  • Intracellular Fluid / metabolism
  • Membrane Potentials / drug effects
  • Membrane Potentials / physiology
  • Patch-Clamp Techniques / methods
  • Peptides, Cyclic / pharmacology
  • Pertussis Toxin / pharmacology
  • Retinal Cone Photoreceptor Cells / cytology*
  • Retinal Cone Photoreceptor Cells / drug effects
  • Retinal Cone Photoreceptor Cells / physiology
  • Somatostatin / pharmacology*

Substances

  • Calcium Channels, L-Type
  • Chelating Agents
  • Enzyme Inhibitors
  • Hormone Antagonists
  • Hormones
  • Peptides, Cyclic
  • 1,2-bis(2-aminophenoxy)ethane N,N,N',N'-tetraacetic acid acetoxymethyl ester
  • Cyanamide
  • Somatostatin
  • Egtazic Acid
  • seglitide
  • Pertussis Toxin
  • Calcium