Soluble epoxide hydrolase gene deletion attenuates renal injury and inflammation with DOCA-salt hypertension

Am J Physiol Renal Physiol. 2009 Sep;297(3):F740-8. doi: 10.1152/ajprenal.00098.2009. Epub 2009 Jun 24.

Abstract

Inhibition of soluble epoxide hydrolase (sEH) has been shown to be renal protective in rat models of salt-sensitive hypertension. Here, we hypothesize that targeted disruption of the sEH gene (Ephx2) prevents both renal inflammation and injury in deoxycorticosterone acetate plus high salt (DOCA-salt) hypertensive mice. Mean arterial blood pressure (MAP) increased significantly in the DOCA-salt groups, and MAP was lower in Ephx2-/- DOCA-salt (129 +/- 3 mmHg) compared with wild-type (WT) DOCA-salt (145 +/- 2 mmHg) mice. Following 21 days of treatment, WT DOCA-salt urinary MCP-1 excretion increased from control and was attenuated in the Ephx2-/- DOCA-salt group. Macrophage infiltration was reduced in Ephx2-/- DOCA-salt compared with WT DOCA-salt mice. Albuminuria increased in WT DOCA-salt (278 +/- 55 microg/day) compared with control (17 +/- 1 microg/day) and was blunted in the Ephx2-/- DOCA-salt mice (97 +/- 23 microg/day). Glomerular nephrin expression demonstrated an inverse relationship with albuminuria. Nephrin immunofluorescence was greater in the Ephx2-/- DOCA-salt group (3.4 +/- 0.3 RFU) compared with WT DOCA-salt group (1.1 +/- 0.07 RFU). Reduction in renal inflammation and injury was also seen in WT DOCA-salt mice treated with a sEH inhibitor {trans-4-[4-(3-adamantan-1-yl-ureido)-cyclohexyloxy]-benzoic acid; tAUCB}, demonstrating that the C-terminal hydrolase domain of the sEH enzyme is responsible for renal protection with DOCA-salt hypertension. These data demonstrate that Ephx2 gene deletion decreases blood pressure, attenuates renal inflammation, and ameliorates glomerular injury in DOCA-salt hypertension.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Albuminuria / enzymology
  • Albuminuria / etiology
  • Albuminuria / prevention & control
  • Animals
  • Benzoates / pharmacology
  • Blood Pressure
  • Chemokine CCL2 / urine
  • Desoxycorticosterone
  • Disease Models, Animal
  • Enzyme Inhibitors / pharmacology
  • Epoxide Hydrolases / antagonists & inhibitors
  • Epoxide Hydrolases / deficiency*
  • Epoxide Hydrolases / genetics
  • Gene Deletion*
  • Hypertension / complications*
  • Hypertension / enzymology
  • Hypertension / etiology
  • Hypertension / physiopathology
  • Kidney Glomerulus / drug effects
  • Kidney Glomerulus / enzymology*
  • Kidney Glomerulus / physiopathology
  • Macrophages / pathology
  • Male
  • Membrane Proteins / metabolism
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Nephritis / enzymology
  • Nephritis / etiology
  • Nephritis / pathology
  • Nephritis / physiopathology
  • Nephritis / prevention & control*
  • Protein Structure, Tertiary
  • Sodium Chloride, Dietary
  • Time Factors
  • Urea / analogs & derivatives
  • Urea / pharmacology

Substances

  • 4-(4-(3-adamantan-1-ylureido)cyclohexyloxy)benzoic acid
  • Benzoates
  • Ccl2 protein, mouse
  • Chemokine CCL2
  • Enzyme Inhibitors
  • Membrane Proteins
  • Sodium Chloride, Dietary
  • nephrin
  • Desoxycorticosterone
  • Urea
  • Epoxide Hydrolases
  • Ephx2 protein, mouse