Regulation of mammary gland branching morphogenesis by EphA2 receptor tyrosine kinase

Mol Biol Cell. 2009 May;20(10):2572-81. doi: 10.1091/mbc.e08-04-0378. Epub 2009 Mar 25.

Abstract

Eph receptor tyrosine kinases, including EphA2, are expressed in the mammary gland. However, their role in mammary gland development remains poorly understood. Using EphA2-deficient animals, we demonstrate for the first time that EphA2 receptor function is required for mammary epithelial growth and branching morphogenesis. Loss of EphA2 decreased penetration of mammary epithelium into fat pad, reduced epithelial proliferation, and inhibited epithelial branching. These defects appear to be intrinsic to loss of EphA2 in epithelium, as transplantation of EphA2-deficient mammary tissue into wild-type recipient stroma recapitulated these defects. In addition, HGF-induced mammary epithelial branching morphogenesis was significantly reduced in EphA2-deficient cells relative to wild-type cells, which correlated with elevated basal RhoA activity. Moreover, inhibition of ROCK kinase activity in EphA2-deficient mammary epithelium rescued branching defects in primary three-dimensional cultures. These results suggest that EphA2 receptor acts as a positive regulator in mammary gland development, functioning downstream of HGF to regulate branching through inhibition of RhoA. Together, these data demonstrate a positive role for EphA2 during normal mammary epithelial proliferation and branching morphogenesis.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Apoptosis / drug effects
  • Cell Proliferation / drug effects
  • Ephrin-A1 / metabolism
  • Epithelial Cells / cytology
  • Epithelial Cells / drug effects
  • Epithelial Cells / enzymology
  • Epithelium / drug effects
  • Epithelium / enzymology
  • Hepatocyte Growth Factor / pharmacology
  • Ligands
  • Mammary Glands, Animal / cytology
  • Mammary Glands, Animal / drug effects
  • Mammary Glands, Animal / enzymology*
  • Mammary Glands, Animal / growth & development*
  • Mice
  • Models, Biological
  • Morphogenesis* / drug effects
  • Receptor, EphA2 / deficiency
  • Receptor, EphA2 / metabolism*
  • rhoA GTP-Binding Protein / metabolism

Substances

  • Ephrin-A1
  • Ligands
  • Hepatocyte Growth Factor
  • Receptor, EphA2
  • rhoA GTP-Binding Protein