Chemical and physical compatibility of levalbuterol inhalation solution concentrate mixed with budesonide, ipratropium bromide, cromolyn sodium, or acetylcysteine sodium

Respir Care. 2008 Dec;53(12):1716-22.

Abstract

Background: Medications are frequently combined in the nebulizer cup, so it is important to determine their chemical and physical compatibility.

Objective: To determine the chemical and physical compatibility of levalbuterol with ipratropium bromide, cromolyn sodium, acetylcysteine sodium, and budesonide.

Methods: We mixed one dose of levalbuterol inhalation solution concentrate (1.25 mg/0.5 mL) with one dose of ipratropium bromide (0.5 mg/2.5 mL), cromolyn sodium (20 mg/2 mL), acetylcysteine sodium (1,000 mg/5 mL), or budesonide (0.5 mg/2 mL). Immediately after mixing the 2 drugs (time zero [T(0)]), and again after 30 min at room temperature (T(30)), we visually inspected the admixtures, measured their pH, and conducted high-pressure liquid chromatography (HPLC).

Results: There was no evidence of physical incompatibility with these drugs combinations. With all the admixtures, both drugs were chemically stable for at least 30-min. Admixture pH had not changed significantly at T(30). Drug recovery was 93.2-102.6% of the initial or control values.

Conclusions: The 2-drug admixtures we studied were compatible for at least 30 min at room temperature.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylcysteine / administration & dosage
  • Acetylcysteine / chemistry*
  • Administration, Inhalation
  • Albuterol / administration & dosage
  • Albuterol / chemistry*
  • Budesonide / administration & dosage
  • Budesonide / chemistry*
  • Cromolyn Sodium / administration & dosage
  • Cromolyn Sodium / chemistry*
  • Drug Incompatibility
  • Drug Stability
  • Drug Therapy, Combination
  • Ipratropium / administration & dosage
  • Ipratropium / chemistry*
  • Respiratory System Agents / administration & dosage
  • Respiratory System Agents / chemistry*
  • Time Factors

Substances

  • Respiratory System Agents
  • Budesonide
  • Ipratropium
  • Cromolyn Sodium
  • Albuterol
  • Acetylcysteine