Ectopic cyclin D1 overexpression increases chemosensitivity but not cell proliferation in multiple myeloma

Int J Oncol. 2008 Dec;33(6):1201-13.

Abstract

We established a myeloma cell line (RPMI8226) with cyclin D1 overexpression in which the transfected cyclin D1 gene was stably expressed. D1 transfectants showed down-regulation of cyclin D2. Cell proliferation analysis did not show any differences among RPMI8226, mock control, and D1 transfectants. The number of S-phase cells increased while the number of G0/G1- and G2/M-phase cells decreased in D1 transfectants, which indicates a prolonged S-phase caused by cyclin D1 transfection. A decreased number of G2/M-phase cells was also detected in myeloma cells of patients with translocation t(11;14)(q13;q32). Western blot analysis revealed an increase in the hyperphosphorylated form of retinoblastoma (Rb) protein in D1 transfectants; however, the expression of p53, p16, Bax, Bad, Bcl-2, and Mcl-1 did not significantly change. Treatment with anti-myeloma drugs (melphalan, dexamethasone, bortezomib and immunomodulatory compounds) induced apoptosis earlier in D1 transfectants compared with RPMI8226 and mock control via the activation of both caspase-8 and -9. However, we could not detect a relationship between cyclin D1 expression and the response to treatment with VAD and bortezomib. Therefore, we assume that high sensitivity to anti-myeloma drugs depends on the duration of the S-phase, but a clinical response might depend on the number of myeloma cells with cyclin D1 overexpression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Antineoplastic Agents* / pharmacology
  • Antineoplastic Agents* / therapeutic use
  • Apoptosis / drug effects*
  • Boronic Acids / therapeutic use
  • Bortezomib
  • Cell Cycle / drug effects*
  • Cell Line, Tumor
  • Cell Proliferation / drug effects*
  • Cyclin D1 / genetics
  • Cyclin D1 / metabolism*
  • Cyclin D2
  • Cyclin-Dependent Kinase Inhibitor p27
  • Cyclins / metabolism
  • Dexamethasone / pharmacology
  • Female
  • Humans
  • Intracellular Signaling Peptides and Proteins / metabolism
  • Male
  • Melphalan / pharmacology
  • Middle Aged
  • Multiple Myeloma / drug therapy*
  • Multiple Myeloma / genetics
  • Multiple Myeloma / metabolism
  • Multiple Myeloma / pathology
  • Phosphorylation
  • Pyrazines / therapeutic use
  • Retinoblastoma Protein / metabolism
  • Thalidomide / pharmacology
  • Time Factors
  • Transfection
  • Up-Regulation
  • Vincristine / therapeutic use

Substances

  • Antineoplastic Agents
  • Boronic Acids
  • CCND1 protein, human
  • CCND2 protein, human
  • CDKN1B protein, human
  • Cyclin D2
  • Cyclins
  • Intracellular Signaling Peptides and Proteins
  • Pyrazines
  • Retinoblastoma Protein
  • Cyclin D1
  • Cyclin-Dependent Kinase Inhibitor p27
  • Thalidomide
  • Vincristine
  • Bortezomib
  • Dexamethasone
  • Melphalan