Converting cell lines representing hematological malignancies from glucocorticoid-resistant to glucocorticoid-sensitive: signaling pathway interactions

Leuk Res. 2009 May;33(5):717-27. doi: 10.1016/j.leukres.2008.10.006. Epub 2008 Nov 13.

Abstract

Mitogen-activated protein kinases (MAPKs), protein kinase A (PKA) and mTOR pathways modulate the apoptotic effects of glucocorticoids (GCs) in human lymphoblastic leukemia CEM cells. We now show that manipulation of these pathways converts several cell lines, representing other lymphoid malignancies, from GC-resistant to GC-sensitive. Basal levels of phosphorylated JNK and ERK were elevated in the GC-resistant cells. Treatments that directly or indirectly reduced phosphorylated JNK and ERK resulted in Dex sensitivity in five resistant lymphoid cell lines. Sensitivity to GC-driven apoptosis correlated with GC-dependent increases in phosphorylated and total glucocorticoid receptor, and in increased levels of the pro-apoptotic protein Bim.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Apoptosis
  • Cell Line, Tumor
  • Dexamethasone / pharmacology*
  • Drug Resistance, Neoplasm
  • Hematologic Neoplasms / enzymology
  • Hematologic Neoplasms / metabolism
  • Hematologic Neoplasms / pathology*
  • Humans
  • Mitogen-Activated Protein Kinases / metabolism
  • Phosphorylation
  • Signal Transduction*

Substances

  • Dexamethasone
  • Mitogen-Activated Protein Kinases