Recent developments in the discovery of selective glucocorticoid receptor modulators (SGRMs)

Curr Top Med Chem. 2008;8(9):750-65. doi: 10.2174/156802608784535048.

Abstract

Steroidal glucocorticoids are widely prescribed for the treatment of a variety of inflammatory and autoimmune diseases. Although they are effective, the side-effects associated with chronic glucocorticoid treatment, such as osteoporosis and hyperglycemia, can severely limit their long-term use. Hence, there is a need to develop new effective anti-inflammatory agents for systemic use which are dissociated from their unwanted side effects.

Publication types

  • Review

MeSH terms

  • Anti-Inflammatory Agents / chemistry*
  • Drug Design
  • Glucocorticoids / chemistry
  • Humans
  • Ligands
  • Receptors, Glucocorticoid / drug effects*
  • Structure-Activity Relationship

Substances

  • Anti-Inflammatory Agents
  • Glucocorticoids
  • Ligands
  • Receptors, Glucocorticoid