Hypocretins and primary headaches: neurobiology and clinical implications

Expert Rev Neurother. 2008 Mar;8(3):409-16. doi: 10.1586/14737175.8.3.409.

Abstract

Hypocretins (or orexins) are two neuropeptides synthesized by neurons located exclusively in the hypothalamus. Hypocretin-containing neurons have widespread projections throughout the CNS; with particularly dense excitatory projections to monoaminergic and serotonergic brainstem centers. The hypocretin system influences a wide range of physiological processes in mammals, such as feeding, arousal, rewards and drug addiction. Recently, a number of studies in experimental animals showed that hypocretins are involved in pain modulation within the CNS, and suggested the presence of a link between these peptides and nociceptive phenomena observed in primary headaches. The aim of this review is to describe and discuss recent studies in humans suggesting a role for the hypocretin neuronal system in cluster headache and chronic migraine.

Publication types

  • Review

MeSH terms

  • Animals
  • Brain Stem / physiology
  • Cluster Headache / physiopathology
  • Headache / physiopathology*
  • Humans
  • Hypothalamus / physiopathology
  • Intracellular Signaling Peptides and Proteins / physiology*
  • Migraine Disorders / physiopathology
  • Neurons / physiology
  • Neuropeptides / physiology*
  • Orexins
  • Pain Threshold / physiology

Substances

  • Intracellular Signaling Peptides and Proteins
  • Neuropeptides
  • Orexins