Inhibition of histone deacetylation protects wildtype but not gelsolin-deficient mice from ischemic brain injury

Exp Neurol. 2008 Apr;210(2):531-42. doi: 10.1016/j.expneurol.2007.11.031. Epub 2007 Dec 23.

Abstract

Acetylation/deactylation of histones is an important mechanism to regulate gene expression and chromatin remodeling. We have previously demonstrated that the HDAC inhibitor trichostatin A (TSA) protects cortical neurons from oxygen/glucose deprivation in vitro which is mediated--at least in part--via the up regulation of gelsolin expression. Here, we demonstrate that TSA treatment dose-dependently enhances histone acetylation in brains of wildtype mice as evidenced by immunoblots of total brain lysates and immunocytochemical staining. Along with increased histone acetylation dose-dependent up regulation of gelsolin protein was observed. Levels of filamentous actin were largely decreased by TSA pre-treatment in brain of wildtype but not gelsolin-deficient mice. When exposed to 1 h filamentous occlusion of the middle cerebral artery followed by reperfusion TSA pre-treated wildtype mice developed significantly smaller cerebral lesion volumes and tended to have improved neurological deficit scores compared to vehicle-treated mice. These protective effects could not be explained by apparent changes in physiological parameters. In contrast to wildtype mice, TSA pre-treatment did not protect gelsolin-deficient mice against MCAo/reperfusion suggesting that enhanced gelsolin expression is an important mechanism by which TSA protects against ischemic brain injury. Our results suggest that HDAC inhibitors such as TSA are a promising therapeutic strategy for reducing brain injury following cerebral ischemia.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylation / drug effects
  • Animals
  • Brain Injuries / etiology*
  • Brain Injuries / metabolism*
  • Brain Injuries / pathology
  • Brain Injuries / prevention & control
  • Brain Ischemia / complications*
  • Brain Ischemia / drug therapy
  • Calcium / metabolism
  • Cells, Cultured
  • Cerebral Cortex / cytology
  • Disease Models, Animal
  • Embryo, Mammalian
  • Enzyme Inhibitors / therapeutic use
  • Gelsolin / deficiency*
  • Glucose / deficiency
  • Histones / metabolism*
  • Hydroxamic Acids / therapeutic use
  • Hypoxia
  • Male
  • Membrane Potential, Mitochondrial / drug effects
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Phosphopyruvate Hydratase / metabolism
  • Rats

Substances

  • Enzyme Inhibitors
  • Gelsolin
  • Histones
  • Hydroxamic Acids
  • trichostatin A
  • Phosphopyruvate Hydratase
  • Glucose
  • Calcium