Reversible inhibition of the fusion activity of measles virus F protein by an engineered intersubunit disulfide bridge

J Virol. 2007 Aug;81(16):8821-6. doi: 10.1128/JVI.00754-07. Epub 2007 Jun 6.

Abstract

In search of target sites for the development of paramyxovirus inhibitors, we have engineered disulfide bridges to introduce covalent links into the prefusion F protein trimer of measles virus. F-Edm-452C/460C, predicted to bridge head and stalk domains of different F monomers, shows a high degree of proteolytic maturation and surface expression, predominantly as stable, dithiothreitol-sensitive trimers, but no fusion activity. Reduction of disulfide bridges partially restores activity. These findings underscore the importance of reversible intersubunit interactions between the stalk and head domains for F activity. Noncovalent small molecules mimicking this behavior may constitute a potent strategy for preventing paramyxovirus entry.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antiviral Agents / pharmacology
  • Biotinylation
  • Chlorocebus aethiops
  • Cysteine / chemistry
  • Cysteine / genetics
  • Disulfides / chemistry*
  • Dithiothreitol / pharmacology
  • Drug Design
  • Measles virus / chemistry*
  • Measles virus / drug effects
  • Membrane Fusion / drug effects*
  • Molecular Sequence Data
  • Mutation
  • Protein Conformation
  • Protein Engineering
  • Streptavidin / chemistry
  • Vero Cells
  • Viral Fusion Proteins / antagonists & inhibitors*
  • Viral Fusion Proteins / chemistry*
  • Viral Fusion Proteins / genetics

Substances

  • Antiviral Agents
  • Disulfides
  • Viral Fusion Proteins
  • Streptavidin
  • Cysteine
  • Dithiothreitol