Improvements in parameters of end-stage liver disease in patients with HIV/HBV-related cirrhosis treated with tenofovir

Antivir Ther. 2007;12(1):119-22.

Abstract

Background: Mortality related to end-stage liver disease is increasing in HIV/hepatitis B virus (HBV)-coinfected patients and effective treatment options are limited. Tenofovir is now widely used in HIV/HBV coinfection and results in significant HBV suppression, in both patients with and patients without lamivudine resistance. The safety and efficacy of tenofovir in HIV/HBV cirrhosis has not been previously described.

Methods: Seven cirrhotic HIV/HBV patients treated with tenofovir were identified within the HIV clinic. Parameters of hepatic function, CD4+ T-cell counts, HBV DNA levels and Child-Pugh Class (C-P-C) were determined before and after addition of tenofovir. All patients had prior lamivudine experience with a median baseline HBV DNA of 6.23 x 10(7) copies/ml.

Results: Four of seven patients were C-P-C -A and hepatitis 'e' antigen (HBeAG) was positive in 4/7 patients. After a median duration of tenofovir of 28 months, all laboratory parameters improved, with significant changes in albumin and prothrombin (PT) (median pre/post-tenofovir: alanine aminotransferase 63/39; bilirubin 26/18; albumin 39/44, P = 0.028; PT 17.5/15, P = 0.018). All three patients with C-P-C -B or -C improved to C-P-C -A, which for one patient enabled removal from the liver transplant waiting list. Three patients lost HBeAG with two anti-HBe seroconversions. Median HBV DNA was suppressed to <35 copies/mi.

Conclusions: This study demonstrates that tenofovir can produce HBV viral suppression, HBeAg seroconversion and improvement in markers of hepatic function in HIV/HBV-coinfected patients with cirrhosis. The potential reversal of end-stage liver disease may provide an important survival benefit in this population.

MeSH terms

  • Adenine / analogs & derivatives*
  • Adenine / therapeutic use
  • CD4 Lymphocyte Count
  • DNA, Viral / blood
  • Follow-Up Studies
  • HIV Infections / complications
  • HIV Infections / drug therapy*
  • HIV Infections / immunology
  • Hepatitis B / blood
  • Hepatitis B / complications
  • Hepatitis B / drug therapy*
  • Hepatitis B / genetics
  • Hepatitis B / immunology
  • Hepatitis B e Antigens / blood
  • Hepatitis B virus / genetics
  • Humans
  • Liver Cirrhosis / complications*
  • Liver Cirrhosis / drug therapy
  • Liver Cirrhosis / pathology
  • Liver Cirrhosis / virology
  • Liver Failure / drug therapy
  • Liver Failure / pathology
  • Liver Failure / virology*
  • Male
  • Middle Aged
  • Organophosphonates / therapeutic use*
  • Reverse Transcriptase Inhibitors / therapeutic use*
  • Severity of Illness Index
  • Tenofovir
  • Time Factors
  • Treatment Outcome
  • Viral Load

Substances

  • DNA, Viral
  • Hepatitis B e Antigens
  • Organophosphonates
  • Reverse Transcriptase Inhibitors
  • Tenofovir
  • Adenine