Iron-regulatory proteins limit hypoxia-inducible factor-2alpha expression in iron deficiency

Nat Struct Mol Biol. 2007 May;14(5):420-6. doi: 10.1038/nsmb1222. Epub 2007 Apr 8.

Abstract

Hypoxia stimulates erythropoiesis, the major iron-utilization pathway. We report the discovery of a conserved, functional iron-responsive element (IRE) in the 5' untranslated region of the messenger RNA encoding endothelial PAS domain protein-1, EPAS1 (also called hypoxia-inducible factor-2alpha, HIF2alpha). Via this IRE, iron regulatory protein binding controls EPAS1 mRNA translation in response to cellular iron availability. Our results uncover a regulatory link that permits feedback control between iron availability and the expression of a key transcription factor promoting iron utilization. They also show that an IRE that is structurally distinct from, for example, the ferritin mRNA IRE and that has been missed by in silico approaches, can mediate mechanistically similar responses.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Basic Helix-Loop-Helix Transcription Factors / genetics*
  • Feedback, Physiological
  • Gene Expression Regulation*
  • HeLa Cells
  • Humans
  • Iron Deficiencies*
  • Iron Metabolism Disorders
  • Iron-Regulatory Proteins / physiology*
  • RNA, Messenger / genetics
  • Response Elements
  • Transcription Factors / genetics

Substances

  • Basic Helix-Loop-Helix Transcription Factors
  • Iron-Regulatory Proteins
  • RNA, Messenger
  • Transcription Factors
  • endothelial PAS domain-containing protein 1