Erythropoietin treatment is associated with more severe thrombocytopenia in patients with chronic hepatitis C undergoing antiviral therapy

Am J Gastroenterol. 2006 Oct;101(10):2275-82. doi: 10.1111/j.1572-0241.2006.00774.x.

Abstract

Background: Erythropoietin (EPO) not only stimulates erythropoiesis but also thrombopoiesis. As pegylated-interferon-alpha(PEG-IFN-alpha)-induced thrombocytopenia may become a limiting factor for continuation of therapy, the present study investigated if EPO can alleviate PEG-IFN-alpha induced thrombocytopenia. Further, we hypothesize that EPO increases platelet reactivity and protease activated receptor 1 (PAR-1) expression during combination antiviral therapy.

Methods: Forty patients with chronic hepatitis C received either 10,000 IU EPO 3 x/week or placebo in a randomized, placebo-controlled, double-blinded fashion for 4 wk and combination antiviral therapy with PEG-IFN-2a and ribavirin.

Results: EPO alleviated the decrease in hemoglobin during combination antiviral therapy with ribavirin (10%vs 20%, p < 0.0001). Platelet counts decreased stronger in EPO than in placebo group on day 28 (p= 0.007). EPO induced a 40% increase in PAR-1 (p < 0.0001), which was accompanied by 100% increase in platelet reactivity (p < 0.0001). PFA-100 platelet plug formation time and PEG-IFN-alpha-induced vWF-increase were not different between study groups.

Conclusions: Treatment with EPO alleviated the decrease in hemoglobin but worsened PEG-IFN-alpha induced thrombocytopenia after the first 4 wk of combination therapy. EPO caused PAR-1 receptor upregulation on platelets, which promoted an increase in platelet reactivity without affecting PFA-100 platelet plug formation time. EPO is not a useful option for short-term support of platelet production during antiviral therapy.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Antiviral Agents / administration & dosage
  • Antiviral Agents / adverse effects*
  • Blood Cell Count
  • Double-Blind Method
  • Drug Therapy, Combination
  • Erythropoietin / administration & dosage
  • Erythropoietin / adverse effects*
  • Female
  • Hepatitis C, Chronic / blood
  • Hepatitis C, Chronic / drug therapy*
  • Humans
  • Interferon alpha-2
  • Interferon-alpha / administration & dosage
  • Interferon-alpha / adverse effects*
  • Male
  • Middle Aged
  • P-Selectin / blood
  • Polyethylene Glycols / administration & dosage
  • Polyethylene Glycols / adverse effects*
  • Receptor, PAR-1 / blood
  • Recombinant Proteins
  • Ribavirin / administration & dosage
  • Ribavirin / adverse effects*
  • Thrombocytopenia / blood
  • Thrombocytopenia / chemically induced*

Substances

  • Antiviral Agents
  • Interferon alpha-2
  • Interferon-alpha
  • P-Selectin
  • Receptor, PAR-1
  • Recombinant Proteins
  • epoetin beta
  • Erythropoietin
  • Polyethylene Glycols
  • Ribavirin
  • peginterferon alfa-2a