Inhibition of cytochrome c oxidase subunit 4 precursor processing by the hypoxia mimic cobalt chloride

Biochem Biophys Res Commun. 2006 Jun 16;344(4):1086-93. doi: 10.1016/j.bbrc.2006.04.014. Epub 2006 Apr 19.

Abstract

Cobalt is often used as a hypoxia mimic in cell culture, because it stabilizes the alpha subunits of the transcription factor, HIF (hypoxia-inducible factor). We have previously shown that HIF stabilization due to a deficiency of the von Hippel Lindau protein (pVHL) in clear cell renal carcinoma (CRCC) was correlated to a down-regulation of oxidative phosphorylation. To better understand this mechanism, we have used CoCl2 in CRCC expressing stably transfected vhl. We show that, in addition to its effect on HIF-alpha subunits, CoCl2 prevented the normal processing of the precursor of cytochrome c oxidase (COX) subunit 4 and induced COX degradation very likely by inhibiting the mitochondrial intermediate peptidase (MIP) that cleaves the COX4 precursor protein. This cobalt-induced MIP inhibition was however not observed in other human mitochondrial precursor sequences as previously predicted from comparison between human and yeast mitochondrial precursor sequences.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Cell Line, Tumor
  • Cobalt / toxicity*
  • Electron Transport Complex IV / antagonists & inhibitors*
  • Electron Transport Complex IV / metabolism*
  • Humans
  • Hypoxia / chemically induced*
  • Hypoxia / enzymology
  • Hypoxia-Inducible Factor 1, alpha Subunit / drug effects
  • Hypoxia-Inducible Factor 1, alpha Subunit / metabolism
  • Metalloendopeptidases / antagonists & inhibitors*
  • Molecular Sequence Data
  • Oxidative Phosphorylation / drug effects
  • Protein Subunits
  • Von Hippel-Lindau Tumor Suppressor Protein / genetics
  • Von Hippel-Lindau Tumor Suppressor Protein / metabolism

Substances

  • Hypoxia-Inducible Factor 1, alpha Subunit
  • Protein Subunits
  • Cobalt
  • Electron Transport Complex IV
  • Von Hippel-Lindau Tumor Suppressor Protein
  • Metalloendopeptidases
  • mitochondrial intermediate peptidase
  • VHL protein, human
  • cobaltous chloride