New approach for high-throughput screening of drug activity on Plasmodium liver stages

Antimicrob Agents Chemother. 2006 Apr;50(4):1586-9. doi: 10.1128/AAC.50.4.1586-1589.2006.

Abstract

Plasmodium liver stages represent potential targets for antimalarial prophylactic drugs. Nevertheless, there is a lack of molecules active on these stages. We have now developed a new approach for the high-throughput screening of drug activity on Plasmodium liver stages in vitro, based on an infrared fluorescence scanning system. This method allowed us to count automatically and rapidly Plasmodium-infected hepatocytes, using different hepatic cells and different Plasmodium species, including Plasmodium falciparum. This new technique is well adapted for high-throughput drug screening and should facilitate the identification of new antimalarial compounds active on Plasmodium liver stages.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antimalarials / pharmacology*
  • Cells, Cultured
  • Hepatocytes / parasitology*
  • Humans
  • Plasmodium / drug effects*

Substances

  • Antimalarials