Population pharmacokinetics as a method to detect variable risperidone exposure in patients suffering from dementia with behavioral disturbances

Am J Geriatr Pharmacother. 2005 Jun;3(2):87-91. doi: 10.1016/j.amjopharm.2005.07.002.

Abstract

Objective: This study was intended to compare the consistency of risperidone exposure in patients who have dementia and behavioral disturbances treated in a psychiatric hospital versus a community care setting.

Methods: Population pharmacokinetic modeling was used to assess the consistency of risperidone exposure in Alzheimer's disease patients with agitation. The ratio of predicted to observed drug concentrations (Cpred/Cobs) derived from this model was used to compare exposure in the inpatient versus long-term/home care settings using both the mean and the variance of this term across groups.

Results: The modeled Cpred/Cobs ratios had a much higher within-subject variance in the inpatients than in the community care patients (117.03% vs 72.35%; P < 0.001). The central tendencies of the Cpred/Cobs ratios across the 2 groups were not significantly different.

Conclusions: Exposure to risperidone was more variable in a psychiatric hospital than in a community care setting. Future research may help to identify the specific contributors to the increased variance observed in this pilot study.

Publication types

  • Comparative Study
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Aged
  • Aged, 80 and over
  • Antipsychotic Agents / blood
  • Antipsychotic Agents / pharmacokinetics*
  • Antipsychotic Agents / therapeutic use*
  • Behavioral Symptoms / drug therapy
  • Clinical Trials as Topic
  • Dementia / drug therapy*
  • Female
  • Home Care Services
  • Hospitalization
  • Humans
  • Male
  • Models, Biological
  • Risperidone / blood
  • Risperidone / pharmacokinetics*
  • Risperidone / therapeutic use*

Substances

  • Antipsychotic Agents
  • Risperidone