A critical review of anagrelide therapy in essential thrombocythemia and related disorders

Leuk Lymphoma. 2005 May;46(5):641-50. doi: 10.1080/10428190400029817.

Abstract

Thrombocytosis is a common clinical problem and it represents either a primary myeloid disorder (a clonal process) or a reactive phenomenon. While reactive thrombocytosis is often inconsequential, clonal thrombocytosis may require cytoreductive therapy to prevent thrombohemorrhagic complications. In this regard, a controlled clinical trial has previously demonstrated the efficacy of hydroxyurea in reducing the risk of thrombosis in high-risk patients with essential thrombocythemia (ET). Despite the absence of similar evidence for clinical benefit, the platelet-lowering agent anagrelide has been widely used in both ET and polycythemia vera (PV) and recent reports of serious side-effects suggest that such practice might be detrimental to patients. In the current review we provide basic drug information as well as a critical assessment of anagrelide treatment in ET and related disorders.

Publication types

  • Review

MeSH terms

  • Clinical Trials as Topic
  • Humans
  • Hydroxyurea / adverse effects
  • Hydroxyurea / therapeutic use
  • Quinazolines / adverse effects
  • Quinazolines / pharmacology
  • Quinazolines / therapeutic use*
  • Thrombocythemia, Essential / drug therapy*
  • Thrombocytosis / drug therapy

Substances

  • Quinazolines
  • anagrelide
  • Hydroxyurea