Anti-Xa activity relates to survival and efficacy in unselected acute coronary syndrome patients treated with enoxaparin

Circulation. 2004 Jul 27;110(4):392-8. doi: 10.1161/01.CIR.0000136830.65073.C7. Epub 2004 Jul 12.

Abstract

Background: Low-molecular-weight heparin (LMWH) is recommended in the treatment of unstable angina (UA)/non-ST-segment-elevation myocardial infarction (NSTEMI), but no relationship has ever been shown between anticoagulation levels obtained with LMWH treatment and clinical outcomes.

Methods and results: In all, 803 consecutive patients with UA/NSTEMI were treated with subcutaneous enoxaparin and were followed up for 30 days. The recommended dose of enoxaparin of 1 mg/kg BID was used throughout the population except when physicians decided on dose reduction because of a history of a recent bleeding event or because of a high bleeding risk. Anti-factor Xa activity was >0.5 IU/mL in 93% of patients; subtherapeutic anti-Xa levels (<0.5 IU/mL) were associated with lower doses of enoxaparin. The 30-day mortality rate was significantly associated with low anti-Xa levels (<0.5 IU/mL), with a >3-fold increase in mortality compared with the patients with anti-Xa levels in the target range of 0.5 to 1.2 IU/mL (P=0.004). Multivariate analysis revealed low anti-Xa activity as an independent predictor of 30-day mortality at least as strong as age, left ventricular function, and renal function. In contrast, anti-Xa activity did not predict major bleeding complications within the range of anti-Xa levels observed in this study.

Conclusions: In this large unselected cohort of patients with UA/NSTEMI patients, low anti-Xa activity on enoxaparin treatment is independently associated with 30-day mortality, which highlights the need for achieving at least the minimum prescribed anti-Xa level of 0.5 IU/mL with enoxaparin whenever possible.

Publication types

  • Clinical Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Angina, Unstable / blood
  • Angina, Unstable / drug therapy*
  • Angina, Unstable / mortality
  • Angina, Unstable / therapy
  • Angioplasty, Balloon, Coronary
  • Anticoagulants / administration & dosage
  • Anticoagulants / adverse effects
  • Anticoagulants / pharmacology
  • Anticoagulants / therapeutic use*
  • Biomarkers
  • Cardiac Catheterization
  • Clopidogrel
  • Cohort Studies
  • Combined Modality Therapy
  • Creatine Kinase / blood
  • Creatine Kinase, MB Form
  • Drug Therapy, Combination
  • Enoxaparin / administration & dosage
  • Enoxaparin / adverse effects
  • Enoxaparin / pharmacology
  • Enoxaparin / therapeutic use*
  • Factor Xa Inhibitors*
  • Female
  • Follow-Up Studies
  • Hemorrhage / chemically induced
  • Hemorrhage / epidemiology
  • Humans
  • Isoenzymes / blood
  • Male
  • Middle Aged
  • Myocardial Infarction / blood
  • Myocardial Infarction / drug therapy*
  • Myocardial Infarction / mortality
  • Myocardial Infarction / therapy
  • Prospective Studies
  • Survival Analysis
  • Ticlopidine / administration & dosage
  • Ticlopidine / analogs & derivatives*
  • Ticlopidine / therapeutic use
  • Treatment Outcome
  • Troponin I / blood

Substances

  • Anticoagulants
  • Biomarkers
  • Enoxaparin
  • Factor Xa Inhibitors
  • Isoenzymes
  • Troponin I
  • Clopidogrel
  • Creatine Kinase
  • Creatine Kinase, MB Form
  • Ticlopidine