T-cadherin is a receptor for hexameric and high-molecular-weight forms of Acrp30/adiponectin

Proc Natl Acad Sci U S A. 2004 Jul 13;101(28):10308-13. doi: 10.1073/pnas.0403382101. Epub 2004 Jun 21.

Abstract

Acrp30/adiponectin is reduced in the serum of obese and diabetic individuals, and the genetic locus of adiponectin is linked to the metabolic syndrome. Recombinant adiponectin, administered to diet-induced obese mice, induced weight loss and improved insulin sensitivity. In muscle and liver, adiponectin stimulates AMP-activated protein kinase activation and fatty acid oxidation. To expression-clone molecules capable of binding adiponectin, we transduced a C2C12 myoblast cDNA retroviral expression library into Ba/F3 cells and panned infected cells on recombinant adiponectin linked to magnetic beads. We identified T-cadherin as a receptor for the hexameric and high-molecular-weight species of adiponectin but not for the trimeric or globular species. Only eukaryotically expressed adiponectin bound to T-cadherin, implying that posttranslational modifications of adiponectin are critical for binding. An adiponectin mutant lacking a conserved N-terminal cysteine residue required for formation of hexamer and high-molecular-weight species did not bind T-cadherin in coimmunoprecipitation studies. Although lacking known cellular functions, T-cadherin is expressed in endothelial and smooth muscle cells, where it is positioned to interact with adiponectin. Because T-cadherin is a glycosylphosphatidylinositol-anchored extracellular protein, it may act as a coreceptor for an as-yet-unidentified signaling receptor through which adiponectin transmits metabolic signals.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adiponectin
  • Adipose Tissue / metabolism
  • Animals
  • CHO Cells
  • Cadherins / genetics
  • Cadherins / metabolism*
  • Cricetinae
  • Flow Cytometry
  • Gene Expression
  • Humans
  • Intercellular Signaling Peptides and Proteins*
  • Kidney / cytology
  • Ligands
  • Magnetics
  • Mice
  • Molecular Weight
  • Myoblasts / cytology
  • Plasmids
  • Protein Binding
  • Proteins / chemistry*
  • Proteins / metabolism*
  • Signal Transduction / physiology

Substances

  • Adiponectin
  • Cadherins
  • H-cadherin
  • Intercellular Signaling Peptides and Proteins
  • Ligands
  • Proteins